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0.014 - 0.037
(7-methoxycoumarin-4-yl)acetyl-Glu-His-Trp-Ser-Tyr-Gly-Leu-Arg-Pro-OH
0.0025
(7-methoxycoumarin-4-yl)acetyl-Gly-Gly-Phe-Ile-Arg-Arg-Ala-Lys-dinitrophenyl
-
recombinant enzyme from E. coli
0.0014
(7-methoxycoumarin-4-yl)acetyl-Gly-Gly-Phe-Leu-Arg-Arg-Ala-Lys-dinitrophenyl
-
recombinant enzyme from E. coli
0.0012 - 0.0057
(7-methoxycoumarin-4-yl)acetyl-Leu-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Lys(Dnp)-OH
0.0045
(o-aminobenzoyl)-AFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0102
(o-aminobenzoyl)-AKPRRPQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 8.0, 37°C, hydrolysis of R-R bond
0.003
(o-aminobenzoyl)-DFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0012
(o-aminobenzoyl)-EFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.001
(o-aminobenzoyl)-FFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0042
(o-aminobenzoyl)-GASPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0166
(o-aminobenzoyl)-GDSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0225
(o-aminobenzoyl)-GESPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.00071
(o-aminobenzoyl)-GFAPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0068
(o-aminobenzoyl)-GFDPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0052
(o-aminobenzoyl)-GFEPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0014
(o-aminobenzoyl)-GFFPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.00072
(o-aminobenzoyl)-GFHPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.00099
(o-aminobenzoyl)-GFIPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.00038
(o-aminobenzoyl)-GFLPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.00027
(o-aminobenzoyl)-GFNPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.006
(o-aminobenzoyl)-GFPPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0149
(o-aminobenzoyl)-GFQPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0053
(o-aminobenzoyl)-GFRPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0012
(o-aminobenzoyl)-GFSAFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0076
(o-aminobenzoyl)-GFSDFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0038
(o-aminobenzoyl)-GFSEFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.00069
(o-aminobenzoyl)-GFSFFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0011
(o-aminobenzoyl)-GFSHFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0016
(o-aminobenzoyl)-GFSLFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0016
(o-aminobenzoyl)-GFSNFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.004
(o-aminobenzoyl)-GFSPARQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.037
(o-aminobenzoyl)-GFSPDRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.018
(o-aminobenzoyl)-GFSPERQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.002
(o-aminobenzoyl)-GFSPFAQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0139
(o-aminobenzoyl)-GFSPFDQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.119
(o-aminobenzoyl)-GFSPFEQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0019
(o-aminobenzoyl)-GFSPFFQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0126
(o-aminobenzoyl)-GFSPFHQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0017
(o-aminobenzoyl)-GFSPFIQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0044
(o-aminobenzoyl)-GFSPFLQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.131
(o-aminobenzoyl)-GFSPFNQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0203
(o-aminobenzoyl)-GFSPFPQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0038
(o-aminobenzoyl)-GFSPFQQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0048
(o-aminobenzoyl)-GFSPFRA-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0012
(o-aminobenzoyl)-GFSPFRE-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.00069
(o-aminobenzoyl)-GFSPFRF-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0005
(o-aminobenzoyl)-GFSPFRI-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.00057
(o-aminobenzoyl)-GFSPFRL-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0018
(o-aminobenzoyl)-GFSPFRN-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0059
(o-aminobenzoyl)-GFSPFRP-(N-(2,4-dinitrophenyl)ethylenediamine)
-
-
0.0022
(o-aminobenzoyl)-GFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.00019
(o-aminobenzoyl)-GFSPFRR-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0043
(o-aminobenzoyl)-GFSPFRS-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.007
(o-aminobenzoyl)-GFSPFSQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0015
(o-aminobenzoyl)-GFSPHRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0085
(o-aminobenzoyl)-GFSPIRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0045
(o-aminobenzoyl)-GFSPLRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.005
(o-aminobenzoyl)-GFSPNRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0043
(o-aminobenzoyl)-GFSPQRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0018
(o-aminobenzoyl)-GFSPRRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0073
(o-aminobenzoyl)-GFSPSRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0075
(o-aminobenzoyl)-GFSQFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0022
(o-aminobenzoyl)-GFSRFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0037
(o-aminobenzoyl)-GFSSFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0012
(o-aminobenzoyl)-GFSXFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0005
(o-aminobenzoyl)-GGFLRRAQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4. 37°C
0.0033
(o-aminobenzoyl)-GGFLRRDQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4. 37°C
0.0019
(o-aminobenzoyl)-GGFLRREQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4. 37°C
0.0007
(o-aminobenzoyl)-GGFLRRFQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4. 37°C
0.0017
(o-aminobenzoyl)-GGFLRRHQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4. 37°C
0.0018
(o-aminobenzoyl)-GGFLRRIQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4. 37°C
0.0007
(o-aminobenzoyl)-GGFLRRLQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4. 37°C
0.0015
(o-aminobenzoyl)-GGFLRRNQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4. 37°C
0.0012
(o-aminobenzoyl)-GGFLRRPQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4. 37°C
0.0023
(o-aminobenzoyl)-GGFLRRRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4. 37°C
0.0022
(o-aminobenzoyl)-GGFLRRV-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4. 37°C
0.0021
(o-aminobenzoyl)-GGFLRRVQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4. 37°C
0.0006
(o-aminobenzoyl)-GGFLRRYQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4. 37°C
0.0048
(o-aminobenzoyl)-GHSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0028
(o-aminobenzoyl)-GISPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0037
(o-aminobenzoyl)-GLSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0045
(o-aminobenzoyl)-GNSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0037
(o-aminobenzoyl)-GPSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0099
(o-aminobenzoyl)-GQSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0036
(o-aminobenzoyl)-GRSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.006
(o-aminobenzoyl)-GSSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0017
(o-aminobenzoyl)-HFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.00016
(o-aminobenzoyl)-IFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.00082
(o-aminobenzoyl)-LFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0071
(o-aminobenzoyl)-NAPRRPQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 8.0, 37°C, hydrolysis of R-R bond
0.00078
(o-aminobenzoyl)-NFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.064
(o-aminobenzoyl)-NKARRPQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 8.0, 37°C, hydrolysis of R-R bond
0.036
(o-aminobenzoyl)-NKPARPQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 8.0, 37°C, hydrolysis of R-R bond
0.015
(o-aminobenzoyl)-NKPRAPQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 8.0, 37°C, hydrolysis of R-R bond
0.0124
(o-aminobenzoyl)-NKPRRAQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 8.0, 37°C, hydrolysis of R-R bond
0.0015
(o-aminobenzoyl)-QFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0015
(o-aminobenzoyl)-RFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.0014
(o-aminobenzoyl)-SFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 7.4, 37°C
0.021
(ortho-aminobenzoyl)-ENKPRRPQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 8.0, 37°C, hydrolysis of R-R bond
0.0028
(ortho-aminobenzoyl)-GGFLPRRPQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 8.0, 37°C, hydrolysis of R-R bond
0.114
(ortho-aminobenzoyl)-KPRRPQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 8.0, 37°C, hydrolysis of R-R bond
0.007
(ortho-aminobenzoyl)-LYENKPRRPQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 8.0, 37°C, hydrolysis of R-R bond
0.0121
(ortho-aminobenzoyl)-NKPRRPQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
pH 8.0, 37°C, hydrolysis of R-R bond
0.0137
2,4-dinitrophenyl-Pro-Leu-Gly-Pro-Trp-D-Lys
-
-
0.0015 - 0.0043
2-aminobenzoyl-GFSPFRQ-(N-2,4-dinitrophenyl)ethylenediamine
0.0123
7-methoxycoumarin-3-carboxylyl-Pro-Leu-Gly-Pro-D-(N6-(2,4-dinitrophenyl))Lys
-
-
0.0082
7-methoxycoumarin-3-carboxylyl-Pro-Leu-Gly-Pro-D-Lys(2,4-dinitrophenyl)
pH and temperature not specified in the publication
0.009 - 0.0343
7-methoxycoumarin-3-carboxylyl-Pro-Leu-Gly-Pro-D-Lys-dinitrophenyl
0.000057 - 0.00127
7-methoxycoumarin-4-acetyl-(L-Ala-L-Lys(2,4-dinitrophenyl))-bradykinin
0.004 - 0.01
7-methoxycoumarin-4-acetyl-Pro-Leu-Gly-Pro-Lys-(2,4-dinitrophenyl)
-
0.00401 - 0.009
7-methoxycoumarin-4-acetyl-Pro-Leu-Gly-Pro-Lys-dinitrophenol
0.000041 - 0.0021
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin
0.0143
Abz-GFSAFRQ-EDDnp
-
pH 7.4, 37°C
0.0012 - 0.0098
Abz-GFSAFRQEDDnp
0.0009
Abz-GFSDFRQ-EDDnp
-
pH 7.4, 37°C
0.0011
Abz-GFSEFRQ-EDDnp
-
pH 7.4, 37°C
0.0021 - 0.0075
Abz-GFSEFRQEDDnp
0.0105
Abz-GFSFFRQ-EDDnp
-
pH 7.4, 37°C
0.0007 - 0.016
Abz-GFSFFRQEDDnp
0.0321
Abz-GFSHFRQ-EDDnp
-
pH 7.4, 37°C
0.0076 - 0.0096
Abz-GFSHFRQEDDnp
0.112
Abz-GFSIFRQ-EDDnp
-
pH 7.4, 37°C
0.0004 - 0.005
Abz-GFSIFRQEDDnp
0.0016 - 0.0102
Abz-GFSLFRQEDDnp
0.0218
Abz-GFSPARQ-EDDnp
-
pH 7.4, 37°C
0.0075
Abz-GFSPDRQ-EDDnp
-
pH 7.4, 37°C
0.0192
Abz-GFSPERQ-EDDnp
-
pH 7.4, 37°C
0.0093
Abz-GFSPFRQ-EDDnp
-
pH 7.4, 37°C
0.0131
Abz-GFSPHRQ-EDDnp
-
pH 7.4, 37°C
0.0062
Abz-GFSPIRQ-EDDnp
-
pH 7.4, 37°C
0.0122
Abz-GFSPLRQ-EDDnp
-
pH 7.4, 37°C
0.0148
Abz-GFSPQRQ-EDDnp
-
pH 7.4, 37°C
0.0213
Abz-GFSPRRQ-EDDnp
-
pH 7.4, 37°C
0.0135
Abz-GFSPSRQ-EDDnp
-
pH 7.4, 37°C
0.0091
Abz-GFSQFRQ-EDDnp
-
pH 7.4, 37°C
0.0012 - 0.0058
Abz-GFSQFRQEDDnp
0.0109
Abz-GFSRFRQ-EDDnp
-
pH 7.4, 37°C
0.0011 - 0.01
Abz-GFSRFRQEDDnp
0.0127
Abz-GFSSFRQ-EDDnp
-
pH 7.4, 37°C
0.0037 - 0.02
Abz-GFSSFRQEDDnp
0.0208
Abz-GFSWFRQ-EDDnp
-
pH 7.4, 37°C
0.0008 - 0.0074
Abz-GFSWFRQEDDnp
0.0009 - 0.011
Abz-GFSyFRQEDDnp
0.067
Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg
-
-
3.1 - 3.45
benzoyl-Gly-Ala-Ala-Gly-p-aminobenzoate
1.54 - 2.5
benzoyl-Gly-Ala-Ala-Leu-p-aminobenzoate
0.058 - 0.83
benzoyl-Gly-Ala-Ala-Phe-p-aminobenzoate
0.37
benzoyl-Gly-Arg-Ala-Ala-Phe-4-aminobenzoate
-
-
-
0.72
benzoyl-Gly-Asp-Ala-Ala-Phe-4-aminobenzoate
-
-
-
1.36 - 2
benzoyl-Gly-Gly-Ala-Phe-p-aminobenzoate
0.24
benzoyl-Gly-Lys-Arg-Ala-Ala-Phe-p-aminobenzoate
-
-
0.16
benzoyl-Gly-Phe-Ala-Ala-Phe-p-aminobenzoate
-
-
0.39 - 0.51
benzoyl-Gly-Phe-Ala-Phe-p-aminobenzoate
0.031
benzoyl-Gly-Phe-Phe-Ala-Ala-Phe-p-aminobenzoate
-
-
0.012 - 0.0161
dinitrophenyl-Pro-Leu-Gly-Pro-Trp-D-Lys
0.048
Gly-Pro-Leu-Gly-Pro-Leu
-
-
0.0149
Gly-Pro-Leu-Gly-Pro-Leu-Gly-Pro-Leu
-
-
0.0135
Gly-Pro-Leu-Gly-Pro-Leu-Gly-Pro-Leu-Gly-Pro-Leu
-
-
0.0154
Gly-Pro-Leu-Gly-Pro-Leu-Gly-Pro-Leu-Gly-Pro-Leu-Gly-Pro-Leu
-
-
0.0026 - 1.64
neurotensin
0.095
pGlu-His-Trp-Ser-Tyr-Gly-Leu-Arg-Pro-Gly-NH2
-
-
0.037
pGlu-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-Leu
-
-
32.5
propionyl-Gly-Ser-Pro-(farnesyl-Cys)-Val-Leu-Met
-
-
0.1 - 0.22
tert-butoxycarbonyl-Phe-Ala-Ala-Phe-p-aminobenzoate
0.06
Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile
-
-
0.038
Tyr-Gly-Gly-Phe-Leu-Arg-Lys-Tyr-Pro
-
-
additional information
additional information
-
kinetics of wild-type and mutant TOP
-
0.014
(7-methoxycoumarin-4-yl)acetyl-Glu-His-Trp-Ser-Tyr-Gly-Leu-Arg-Pro-OH
-
mutant Y605FY612F, 23°C, pH 7.8
0.024
(7-methoxycoumarin-4-yl)acetyl-Glu-His-Trp-Ser-Tyr-Gly-Leu-Arg-Pro-OH
-
wild-type, 23°C, pH 7.8
0.034
(7-methoxycoumarin-4-yl)acetyl-Glu-His-Trp-Ser-Tyr-Gly-Leu-Arg-Pro-OH
-
mutant Y612F, 23°C, pH 7.8
0.037
(7-methoxycoumarin-4-yl)acetyl-Glu-His-Trp-Ser-Tyr-Gly-Leu-Arg-Pro-OH
-
mutant Y605F, 23°C, pH 7.8
0.0012
(7-methoxycoumarin-4-yl)acetyl-Leu-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Lys(Dnp)-OH
-
wild-type, 23°C, pH 7.8
0.0025
(7-methoxycoumarin-4-yl)acetyl-Leu-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Lys(Dnp)-OH
-
mutant G599A, 23°C, pH 7.8
0.0026
(7-methoxycoumarin-4-yl)acetyl-Leu-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Lys(Dnp)-OH
-
mutant G604A, 23°C, pH 7.8
0.0026
(7-methoxycoumarin-4-yl)acetyl-Leu-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Lys(Dnp)-OH
-
mutant Y612F, 23°C, pH 7.8
0.0029
(7-methoxycoumarin-4-yl)acetyl-Leu-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Lys(Dnp)-OH
-
mutant G603A, 23°C, pH 7.8
0.0029
(7-methoxycoumarin-4-yl)acetyl-Leu-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Lys(Dnp)-OH
-
mutant G603P, 23°C, pH 7.8
0.0031
(7-methoxycoumarin-4-yl)acetyl-Leu-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Lys(Dnp)-OH
-
mutant Y605FY612F, 23°C, pH 7.8
0.0042
(7-methoxycoumarin-4-yl)acetyl-Leu-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Lys(Dnp)-OH
-
mutant Y605F, 23°C, pH 7.8
0.005
(7-methoxycoumarin-4-yl)acetyl-Leu-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Lys(Dnp)-OH
-
mutant G611A, 23°C, pH 7.8
0.0057
(7-methoxycoumarin-4-yl)acetyl-Leu-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Lys(Dnp)-OH
-
mutant G603A/G604A, 23°C, pH 7.8
0.0015
2-aminobenzoyl-GFSPFRQ-(N-2,4-dinitrophenyl)ethylenediamine
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605F
0.0022
2-aminobenzoyl-GFSPFRQ-(N-2,4-dinitrophenyl)ethylenediamine
-
pH 7.4, 37°C, recombinant GST-tagged wild-type enzyme
0.0043
2-aminobenzoyl-GFSPFRQ-(N-2,4-dinitrophenyl)ethylenediamine
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605A
0.009
7-methoxycoumarin-3-carboxylyl-Pro-Leu-Gly-Pro-D-Lys-dinitrophenyl
-
-
0.023
7-methoxycoumarin-3-carboxylyl-Pro-Leu-Gly-Pro-D-Lys-dinitrophenyl
-
-
0.0343
7-methoxycoumarin-3-carboxylyl-Pro-Leu-Gly-Pro-D-Lys-dinitrophenyl
-
recombinant enzyme from E. coli
0.000057
7-methoxycoumarin-4-acetyl-(L-Ala-L-Lys(2,4-dinitrophenyl))-bradykinin
pH 7.8, 23°C
0.00013
7-methoxycoumarin-4-acetyl-(L-Ala-L-Lys(2,4-dinitrophenyl))-bradykinin
pH 7.8, 23°C, presence of 1.5 M urea
0.00048
7-methoxycoumarin-4-acetyl-(L-Ala-L-Lys(2,4-dinitrophenyl))-bradykinin
pH 7.8, 23°C, presence of 2.5 M urea
0.00127
7-methoxycoumarin-4-acetyl-(L-Ala-L-Lys(2,4-dinitrophenyl))-bradykinin
pH 7.8, 23°C, presence of 3.5 M urea
0.004
7-methoxycoumarin-4-acetyl-Pro-Leu-Gly-Pro-Lys-(2,4-dinitrophenyl)
pH 7.0, with Ca2+
-
0.0046
7-methoxycoumarin-4-acetyl-Pro-Leu-Gly-Pro-Lys-(2,4-dinitrophenyl)
pH 7.8, wild-type enzyme
-
0.0051
7-methoxycoumarin-4-acetyl-Pro-Leu-Gly-Pro-Lys-(2,4-dinitrophenyl)
pH 7.8, mutant enzyme Y612F
-
0.01
7-methoxycoumarin-4-acetyl-Pro-Leu-Gly-Pro-Lys-(2,4-dinitrophenyl)
pH 7.0, without Ca2+ or at pH 5.8 with or without Ca2+
-
0.00401
7-methoxycoumarin-4-acetyl-Pro-Leu-Gly-Pro-Lys-dinitrophenol
-
mutant G603A, 23°C, pH 7.8
0.00408
7-methoxycoumarin-4-acetyl-Pro-Leu-Gly-Pro-Lys-dinitrophenol
-
mutant G599A, 23°C, pH 7.8
0.00543
7-methoxycoumarin-4-acetyl-Pro-Leu-Gly-Pro-Lys-dinitrophenol
-
mutant G603A/G604A, 23°C, pH 7.8
0.00643
7-methoxycoumarin-4-acetyl-Pro-Leu-Gly-Pro-Lys-dinitrophenol
-
mutant G603P, 23°C, pH 7.8
0.0067
7-methoxycoumarin-4-acetyl-Pro-Leu-Gly-Pro-Lys-dinitrophenol
-
mutant G611A, 23°C, pH 7.8
0.00788
7-methoxycoumarin-4-acetyl-Pro-Leu-Gly-Pro-Lys-dinitrophenol
-
wild-type, 23°C, pH 7.8
0.0081
7-methoxycoumarin-4-acetyl-Pro-Leu-Gly-Pro-Lys-dinitrophenol
-
mutant Y605FY612F, 23°C, pH 7.8
0.0082
7-methoxycoumarin-4-acetyl-Pro-Leu-Gly-Pro-Lys-dinitrophenol
-
mutant Y605F, 23°C, pH 7.8
0.00825
7-methoxycoumarin-4-acetyl-Pro-Leu-Gly-Pro-Lys-dinitrophenol
-
mutant G604A, 23°C, pH 7.8
0.009
7-methoxycoumarin-4-acetyl-Pro-Leu-Gly-Pro-Lys-dinitrophenol
-
mutant Y612F, 23°C, pH 7.8
0.000041
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin
-
mutant G603A/G604A, 23°C, pH 7.8
0.000054
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin
-
mutant G603A, 23°C, pH 7.8
0.000057
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin
-
wild-type, 23°C, pH 7.8
0.00008
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin
-
mutant Y605F, 23°C, pH 7.8
0.00009
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin
-
mutant G604A, 23°C, pH 7.8
0.000129
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin
-
mutant G599A, 23°C, pH 7.8
0.000136
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin
-
mutant G611A, 23°C, pH 7.8
0.00051
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin
-
mutant Y605FY612F, 23°C, pH 7.8
0.00057
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin
-
mutant Y612F, 23°C, pH 7.8
0.0021
7-methoxycoumarin-4-acetyl-[Ala7, Lys(dinitrophenol)9]-bradykinin
-
mutant G603P, 23°C, pH 7.8
0.0012
Abz-GFSAFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged wild-type enzyme
0.0047
Abz-GFSAFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605F
0.0098
Abz-GFSAFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605A
0.0021
Abz-GFSEFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605F
0.003
Abz-GFSEFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605A
0.0075
Abz-GFSEFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged wild-type enzyme
0.0007
Abz-GFSFFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged wild-type enzyme
0.0033
Abz-GFSFFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605F
0.016
Abz-GFSFFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605A
0.0076
Abz-GFSHFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged wild-type enzyme
0.0086
Abz-GFSHFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605F
0.0096
Abz-GFSHFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605A
0.0004
Abz-GFSIFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged wild-type enzyme
0.0014
Abz-GFSIFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605F
0.005
Abz-GFSIFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605A
0.0016
Abz-GFSLFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged wild-type enzyme
0.0032
Abz-GFSLFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605F
0.0102
Abz-GFSLFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605A
0.0012
Abz-GFSQFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged wild-type enzyme
0.0054
Abz-GFSQFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605F
0.0058
Abz-GFSQFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605A
0.0011
Abz-GFSRFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged wild-type enzyme
0.0044
Abz-GFSRFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605F
0.01
Abz-GFSRFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605A
0.0037
Abz-GFSSFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged wild-type enzyme
0.0047
Abz-GFSSFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605F
0.02
Abz-GFSSFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605A
0.0008
Abz-GFSWFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged wild-type enzyme
0.0015
Abz-GFSWFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605F
0.0074
Abz-GFSWFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605A
0.0009
Abz-GFSyFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged wild-type enzyme
0.0023
Abz-GFSyFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605F
0.011
Abz-GFSyFRQEDDnp
-
pH 7.4, 37°C, recombinant GST-tagged mutant Y605A
3.1
benzoyl-Gly-Ala-Ala-Gly-p-aminobenzoate
-
-
3.45
benzoyl-Gly-Ala-Ala-Gly-p-aminobenzoate
-
-
1.54
benzoyl-Gly-Ala-Ala-Leu-p-aminobenzoate
-
-
2.5
benzoyl-Gly-Ala-Ala-Leu-p-aminobenzoate
-
-
0.058
benzoyl-Gly-Ala-Ala-Phe-p-aminobenzoate
-
-
0.49
benzoyl-Gly-Ala-Ala-Phe-p-aminobenzoate
-
-
0.83
benzoyl-Gly-Ala-Ala-Phe-p-aminobenzoate
-
-
1.36
benzoyl-Gly-Gly-Ala-Phe-p-aminobenzoate
-
-
2
benzoyl-Gly-Gly-Ala-Phe-p-aminobenzoate
-
-
0.39
benzoyl-Gly-Phe-Ala-Phe-p-aminobenzoate
-
-
0.51
benzoyl-Gly-Phe-Ala-Phe-p-aminobenzoate
-
-
0.012
dinitrophenyl-Pro-Leu-Gly-Pro-Trp-D-Lys
-
-
0.0133
dinitrophenyl-Pro-Leu-Gly-Pro-Trp-D-Lys
-
-
0.0161
dinitrophenyl-Pro-Leu-Gly-Pro-Trp-D-Lys
-
recombinant enzyme from E. coli
0.0026
neurotensin
-
recombinant wild-type enzyme, pH 7.5, 37°C
0.0033
neurotensin
-
recombinant mutant E469R/R498T, pH 7.5, 37°C
0.1
tert-butoxycarbonyl-Phe-Ala-Ala-Phe-p-aminobenzoate
-
-
0.22
tert-butoxycarbonyl-Phe-Ala-Ala-Phe-p-aminobenzoate
-
-