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3.4.24.82: ADAMTS-4 endopeptidase

This is an abbreviated version!
For detailed information about ADAMTS-4 endopeptidase, go to the full flat file.

Word Map on EC 3.4.24.82

Reaction

Glutamyl endopeptidase; bonds cleaved include -Thr-Glu-Gly-Glu373-/-Ala-Arg-Gly-Ser- in the interglobular domain of mammalian aggrecan =

Synonyms

a disintegrin and metalloprotease with thrombospondin motifs-4, a disintegrin and metalloproteinase with thrombospondin motif, a disintegrin and metalloproteinase with thrombospondin motifs 4, a disintegrin and metalloproteinase with thrombospondin motifs-4, a disintegrin and metalloproteinase with thrombospondin-1-like motifs, a disintegrin-like and metalloproteinase with thrombospondin motifs-4, a disintegrin-like and metalloproteinase with thrombospondin type-1 motifs-4, ADAMTS 4, ADAMTS-1, ADAMTS-4, ADAMTS-4 [a disintegrin and metalloproteinase with thrombospondin motifs-4], ADAMTS-4-2, ADAMTS4, agg-1, aggrecanase, aggrecanase 1, aggrecanase-1, disintegrin and metalloproteinase with thrombospondin motif 4, TS-4

ECTree

     3 Hydrolases
         3.4 Acting on peptide bonds (peptidases)
             3.4.24 Metalloendopeptidases
                3.4.24.82 ADAMTS-4 endopeptidase

IC50 Value

IC50 Value on EC 3.4.24.82 - ADAMTS-4 endopeptidase

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IC50 VALUE [mM]
INHIBITOR
ORGANISM
UNIPROT
COMMENTARY hide
LITERATURE
IMAGE
0.0028
(2R)-2-(biphenyl-4-ylsulfonyl)-3-(1H-indol-2-yl)propanoic acid
Rattus norvegicus
-
IC50: 0.0028 mM
0.0043
(2R)-2-(biphenyl-4-ylsulfonyl)-3-phenylpropanoic acid
Rattus norvegicus
-
IC50: 0.0043 mM
0.0011
(2R)-2-(biphenyl-4-ylsulfonyl)pentanedioic acid
Rattus norvegicus
-
IC50: 0.0011 mM
0.0055
(2R)-2-(biphenyl-4-ylsulfonyl)propanoic acid
Rattus norvegicus
-
IC50: 0.0055 mM
0.02
(2R)-2-([[3'-(acetylamino)biphenyl-4-yl]sulfonyl]amino)-3-methylbutanoic acid
Homo sapiens
-
IC50 around 0.02 mM, pH and temperature not specified in the publication
0.0072
(2R)-2-([[3'-(aminomethyl)biphenyl-4-yl]sulfonyl]amino)-3-methylbutanoic acid
Homo sapiens
-
pH and temperature not specified in the publication
0.0021
(2R)-2-([[3'-(hydroxymethyl)biphenyl-4-yl]sulfonyl]amino)-3-methylbutanoic acid
Homo sapiens
-
pH and temperature not specified in the publication
0.1
(2R)-2-([[4'-(acetylamino)biphenyl-4-yl]sulfonyl]amino)-3-methylbutanoic acid
Homo sapiens
-
IC50 around 0.1 mM, pH and temperature not specified in the publication
0.00042 - 0.0041
(2R)-2-([[4'-(carbamoyloxy)biphenyl-4-yl]sulfonyl]amino)-3-methylbutanoic acid
0.015
(2R)-2-([[4'-(hydroxymethyl)biphenyl-4-yl]sulfonyl]amino)-3-methylbutanoic acid
Homo sapiens
-
pH and temperature not specified in the publication
0.003
(2R)-2-[(biphenyl-4-ylsulfonyl)amino]-3-methylbutanoic acid
Homo sapiens
-
pH and temperature not specified in the publication
0.0084
(2R)-2-[[(3'-carbamoylbiphenyl-4-yl)sulfonyl]amino]-3-methylbutanoic acid
Homo sapiens
-
pH and temperature not specified in the publication
0.04
(2R)-2-[[(3'-cyanobiphenyl-4-yl)sulfonyl]amino]-3-methylbutanoic acid
Homo sapiens
-
pH and temperature not specified in the publication
0.009
(2R)-2-[[(3'-hydroxybiphenyl-4-yl)sulfonyl]amino]-3-methylbutanoic acid
Homo sapiens
-
pH and temperature not specified in the publication
0.0046
(2R)-2-[[(4'-hydroxybiphenyl-4-yl)sulfonyl]amino]-3-methylbutanoic acid
Homo sapiens
-
pH and temperature not specified in the publication
0.05
(2R)-3-methyl-2-[([4'-[(methylcarbamoyl)oxy]biphenyl-4-yl]sulfonyl)amino]butanoic acid
Homo sapiens
-
IC50 around 0.05 mM, pH and temperature not specified in the publication
0.000065
(2R)-N4-hydroxy-2-(3-hydroxybenzyl)-N1-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]butanediamide
Homo sapiens
-
pH 7.5, 37°C
0.0000011
(2R,5R)-1-([4-[(2,4-dichlorobenzyl)oxy]phenyl]sulfonyl)-N,5-dihydroxy-3,3-dimethylpiperidine-2-carboxamide
Homo sapiens
-
37°C, pH and temperature not specified in the publication
0.000145
(2R,5R)-1-([4-[(5-fluoro-2-methylbenzyl)oxy]phenyl]sulfonyl)-N,5-dihydroxypiperidine-2-carboxamide
Homo sapiens
-
IC50: 145 nM
0.0000021
(2R,5R)-N,5-dihydroxy-1-([4-[(2,4-dichlorobenzyl)oxy]phenyl]sulfonyl)piperidine-2-carboxamide
Homo sapiens
-
IC50: 2.1 nM
0.000016
(2R,5R)-N,5-dihydroxy-1-([4-[(2-bromobenzyl)oxy]phenyl]sulfonyl)piperidine-2-carboxamide
Homo sapiens
-
IC50: 16 nM
0.0000005
(2R,5R)-N,5-dihydroxy-1-([4-[(2-chloro-4-fluorobenzyl)oxy]phenyl]sulfonyl)piperidine-2-carboxamide
Homo sapiens
-
IC50: 0.5 nM
0.000067
(2R,5R)-N,5-dihydroxy-1-([4-[(2-ethylbenzyl)oxy]phenyl]sulfonyl)piperidine-2-carboxamide
Homo sapiens
-
IC50: 67 nM
0.0000039
(2R,5R)-N,5-dihydroxy-1-([4-[(2-methyl-3-fluorobenzyl)oxy]phenyl]sulfonyl)piperidine-2-carboxamide
Homo sapiens
-
IC50: 3.9 nM
0.0000027
(2R,5R)-N,5-dihydroxy-1-([4-[(2-methyl-4-fluorobenzyl)oxy]phenyl]sulfonyl)piperidine-2-carboxamide
Homo sapiens
-
IC50: 2.7 nM
0.00004
(2R,5R)-N,5-dihydroxy-1-([4-[(2-methyl-5-fluorobenzyl)oxy]phenyl]sulfonyl)piperidine-2-carboxamide
Homo sapiens
-
IC50: 40 nM
0.000038
(2R,5R)-N,5-dihydroxy-1-([4-[(2-methylbenzyl)oxy]phenyl]sulfonyl)piperidine-2-carboxamide
Homo sapiens
-
IC50: 38 nM
0.0001
(2R,5R)-N,5-dihydroxy-1-([4-[(3-methylbenzyl)oxy]phenyl]sulfonyl)piperidine-2-carboxamide
Homo sapiens
-
IC50: 100 nM
0.0001
(2R,5R)-N,5-dihydroxy-1-([4-[(4-bromobenzyl)oxy]phenyl]sulfonyl)piperidine-2-carboxamide
Homo sapiens
-
IC50: 100 nM
0.000018
(2R,5R)-N,5-dihydroxy-1-[[4-(2-chloropyridin-4-ylmethoxy)phenyl]sulfonyl]piperidine-2-carboxamide
Homo sapiens
-
IC50: 18 nM
0.000091
(2R,5R)-N,5-dihydroxy-1-[[4-(2-methylpyridin-3-ylmethoxy)phenyl]sulfonyl]piperidine-2-carboxamide
Homo sapiens
-
IC50: 91 nM
0.0001
(2R,5R)-N,5-dihydroxy-1-[[4-(isoquinolin-4-ylmethoxy)phenyl]sulfonyl]piperidine-2-carboxamide
Homo sapiens
-
IC50: 100 nM
0.000015
(2R,5R)-N,5-dihydroxy-1-[[4-(quinolin-4-ylmethoxy)phenyl]sulfonyl]piperidine-2-carboxamide
Homo sapiens
-
IC50: 15 nM
0.000003
(3R)-N2-(cyclopropylmethyl)-N1-hydroxy-3-(3-hydroxybenzyl)-N4-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-L-aspartamide
Homo sapiens
-
pH 7.5, 37°C
0.00018
(R)-2-(3-fluoro-4'-((5-oxo-5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl)biphenyl-4-ylsulfonamido)-3-methylbutanoic acid
Mus musculus
-
0.0002
(R)-2-(4'-((2,8-bis(trifluoromethyl)quinolin-4-yloxy)methyl)biphenyl-4-ylsulfonamido)-3-methylbutanoic acid
Mus musculus
-
0.0049
(R)-2-(4'-((3-(dimethylamino)phenoxy)methyl)biphenyl-4-ylsulfonamido)-3-methylbutanoic acid
Mus musculus
-
0.001
(R)-2-(4'-((3-acetylphenoxy)methyl)biphenyl-4-ylsulfonamido)-3-methylbutanoic acid
Mus musculus
-
0.00023
(R)-2-(4'-((3-benzoylphenoxy)methyl)biphenyl-4-ylsulfonamido)-3-methylbutanoic acid
Mus musculus
-
0.0012
(R)-2-(4'-((3-fluorophenoxy)methyl)biphenyl-4-ylsulfonamido)-3-methylbutanoic acid
Mus musculus
-
0.0011
(R)-2-(4'-((3-hydroxyphenoxy)methyl)biphenyl-4-ylsulfonamido)-3-methylbutanoic acid
Mus musculus
-
0.0018
(R)-2-(4'-((3-methoxyphenoxy)methyl)biphenyl-4-ylsulfonamido)-3-methylbutanoic acid
Mus musculus
-
0.00008
(R)-2-(4'-((4-(4-fluorobenzoyl)phenoxy)methyl)biphenyl-4-ylsulfonamido)-3-methylbutanoic acid
Mus musculus
-
0.00009
(R)-2-(4'-((4-(cyclohexanecarbonyl)phenoxy)methyl)biphenyl-4-ylsulfonamido)-3-methylbutanoic acid
Mus musculus
-
0.00059
(R)-2-(4'-((4-(tert-butoxycarbonylamino)phenoxy)methyl)biphenyl-4-ylsulfonamido)-3-methylbutanoic acid
Mus musculus
-
0.00043
(R)-2-(4'-((4-acetylphenoxy)methyl)biphenyl-4-ylsulfonamido)-3-methylbutanoic acid
Mus musculus
-
0.0017
(R)-2-(4'-((4-fluorophenoxy)methyl)biphenyl-4-ylsulfonamido)-3-methylbutanoic acid
Mus musculus
-
0.0001
(R)-2-(4'-((4-isobutyrylphenoxy)methyl)biphenyl-4-ylsulfonamido)-3-methylbutanoic acid
Mus musculus
-
0.0016
(R)-2-(4'-((4-methoxyphenoxy)methyl)biphenyl-4-ylsulfonamido)-3-methylbutanoic acid
Mus musculus
-
0.0002
(R)-3-methyl-2-(4'-((3-methylquinolin-2-yloxy)methyl)biphenyl-4-ylsulfonamido)butanoic acid
Mus musculus
-
0.00073
(R)-3-methyl-2-(4'-((4-(6-methylpyridin-2-yloxy)phenoxy)methyl)biphenyl-4-ylsulfonamido)butanoic acid
Mus musculus
-
0.0052
(R)-3-methyl-2-(4'-((4-(morpholine-4-carbonyl)phenoxy)methyl)biphenyl-4-ylsulfonamido)butanoic acid
Mus musculus
-
0.006
(R)-3-methyl-2-(4'-((4-(morpholinomethyl)phenoxy)methyl)biphenyl-4-ylsulfonamido)butanoic acid
Mus musculus
-
0.0009
(R)-3-methyl-2-(4'-((4-(pyridin-2-yloxy)phenoxy)methyl)biphenyl-4-ylsulfonamido)butanoic acid
Mus musculus
-
0.0019
(R)-3-methyl-2-(4'-((4-(pyrrolidine-1-carbonyl)phenoxy)methyl)biphenyl-4-ylsulfonamido)butanoic acid
Mus musculus
-
0.0004
(R)-3-methyl-2-(4'-((4-phenoxyphenoxy)methyl)biphenyl-4-ylsulfonamido)butanoic acid
Mus musculus
-
0.0008
(R)-3-methyl-2-(4'-((5-(trifluoromethyl)pyridin-2-yloxy)methyl)biphenyl-4-ylsulfonamido)butanoic acid
Mus musculus
-
0.02
(R)-3-methyl-2-(4'-((5-oxo-5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl)-3-(trifluoromethoxy)biphenyl-4-ylsulfonamido)butanoic acid
Mus musculus
-
0.0032
(R)-3-methyl-2-(4'-((5-oxo-5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl)-3-(trifluoromethyl)biphenyl-4-ylsulfonamido)butanoic acid
Mus musculus
-
0.00023
(R)-3-methyl-2-(4'-((5-oxo-5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl)biphenyl-4-ylsulfonamido)butanoic acid
Mus musculus
-
0.0004
(R)-3-methyl-2-(4'-((quinolin-2-yloxy)methyl)biphenyl-4-ylsulfonamido)butanoic acid
Mus musculus
-
0.015
2-[4-(benzyloxy)phenyl]-2,3-dihydro-1-oxo-1H-pyrrolo[3,4-c]quinoline-4-carboxylate
Homo sapiens
-
37°C, pH and temperature not specified in the publication
0.00021
2-[4-(benzyloxy)phenyl]-2,3-dihydro-N-hydroxy-1-oxo-1H-pyrrolo[3,4-c]quinoline-4-carboxamide
Homo sapiens
-
37°C, pH and temperature not specified in the publication
0.1
3-[(biphenyl-4-ylsulfonyl)amino]-4-methylpentanoic acid
Rattus norvegicus
-
IC50: 0.1 mM
0.022
3-[[(4'-[[(1R)-1-carboxy-2-methylpropyl]sulfamoyl]biphenyl-4-yl)oxy]methyl]benzoic acid
Homo sapiens
-
IC50 around 0.022 mM, pH and temperature not specified in the publication
0.00012
AG3340
Bos taurus
-
non-peptidomimetric hydroxamate matrix metalloproteinase inhibitor, IC50: 120 nM
0.0000789
antibody 237-53
Homo sapiens
at pH and 37°C
-
0.00015
BB-16
Bos taurus
-
peptidomimetric hydroxamate, synthetic inhibitor originally targeted for matrix metalloproteinases, IC50: 150 nM
0.00017
C-terminal 40-kDa fibronectin fragment
Bos taurus
-
wild type enzyme IC50: 170 nM, complete inhibition at 750 nM
-
0.00001
DPC
Bos taurus
-
non-peptidomimetric hydroxamate matrix metalloproteinase inhibitor, IC50: 10 nM
0.00011
fibronectin
-
0.000079 - 0.00021
marimastat
0.1
N-(biphenyl-3-ylsulfonyl)-D-valine
Rattus norvegicus
-
IC50: 0.1 mM
0.003
N-(biphenyl-4-ylsulfonyl)-D-valine
Rattus norvegicus
-
IC50: 0.003 mM
0.1
N-(biphenyl-4-ylsulfonyl)-L-valine
Rattus norvegicus
-
IC50: 0.1 mM
0.012
N-(biphenyl-4-ylsulfonyl)-N-(pyridin-3-ylmethyl)-D-valine
Rattus norvegicus
-
IC50: 0.012 mM
0.0016
N-(biphenyl-4-ylsulfonyl)-N-methyl-D-valine
Rattus norvegicus
-
IC50: 0.0016 mM
0.2
N-([3'-[(acetylamino)methyl]biphenyl-4-yl]sulfonyl)-D-valine
Homo sapiens
-
IC50 above 0.2 mM, pH and temperature not specified in the publication
0.0075
N-([4'-[(1-benzofuran-2-ylcarbonyl)amino]biphenyl-4-yl]sulfonyl)-D-valine
Rattus norvegicus
-
IC50: 0.0075 mM
0.00035
N-([4'-[(1-benzofuran-2-ylcarbonyl)oxy]biphenyl-4-yl]sulfonyl)-D-valine
Rattus norvegicus
-
IC50: 0.00035 mM
0.015
N-([4'-[(2-cyanobenzyl)oxy]biphenyl-4-yl]sulfonyl)-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.0024
N-([4'-[(2-methylpyridin-4-yl)methoxy]biphenyl-4-yl]sulfonyl)-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.0005
N-([4'-[(2-methylquinolin-4-yl)methoxy]biphenyl-4-yl]sulfonyl)-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.00042
N-([4'-[(3-bromobenzyl)oxy]biphenyl-4-yl]sulfonyl)-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.0004
N-([4'-[(3-chlorobenzyl)oxy]biphenyl-4-yl]sulfonyl)-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.0008
N-([4'-[(3-cyanobenzyl)oxy]biphenyl-4-yl]sulfonyl)-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.0026
N-([4'-[(3-fluorobenzyl)oxy]biphenyl-4-yl]sulfonyl)-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.0037
N-([4'-[(3-hydroxybenzyl)oxy]biphenyl-4-yl]sulfonyl)-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.00054
N-([4'-[(3-nitrobenzyl)oxy]biphenyl-4-yl]sulfonyl)-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.0014
N-([4'-[(4-cyanobenzyl)oxy]biphenyl-4-yl]sulfonyl)-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.1
N-([4'-[(benzoylamino)methyl]biphenyl-4-yl]sulfonyl)-D-valine
Homo sapiens
-
IC50 around 0.1 mM, pH and temperature not specified in the publication
0.025
N-([4'-[(benzylcarbamoyl)oxy]biphenyl-4-yl]sulfonyl)-D-valine
Homo sapiens
-
IC50 around 0.025 mM, pH and temperature not specified in the publication
0.0116
N-([4'-[(furan-2-yloxy)carbonyl]biphenyl-4-yl]sulfonyl)-D-valine
Rattus norvegicus
-
IC50: 0.0116 mM
0.0056
N-([4'-[(phenylcarbamoyl)oxy]biphenyl-4-yl]sulfonyl)-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.0082
N-([4'-[(phenylsulfonyl)oxy]biphenyl-4-yl]sulfonyl)-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.0004
N-([4'-[(Z)-2-(1-benzofuran-2-yl)ethenyl]biphenyl-4-yl]sulfonyl)-D-valine
Rattus norvegicus
-
IC50: 0.0004 mM
0.0038
N-([4'-[2-(1-benzofuran-2-yl)-2-oxoethyl]biphenyl-4-yl]sulfonyl)-D-valine
Rattus norvegicus
-
IC50: 0.0038 mM
0.05
N-[(2'-aminobiphenyl-4-yl)sulfonyl]-D-valine
Rattus norvegicus
-
IC50: 0.05 mM
0.02
N-[(2'-hydroxybiphenyl-4-yl)sulfonyl]-D-valine
Rattus norvegicus
-
IC50: 0.02 mM
0.03
N-[(2-aminobiphenyl-4-yl)sulfonyl]-D-valine
Rattus norvegicus
-
IC50: 0.03 mM
0.009
N-[(3'-hydroxybiphenyl-4-yl)sulfonyl]-D-valine
Rattus norvegicus
-
IC50: 0.009 mM
0.0046
N-[(4'-hydroxybiphenyl-4-yl)sulfonyl]-D-valine
Rattus norvegicus
-
IC50: 0.0046 mM
0.0132
N-[(4'-phenoxybiphenyl-4-yl)sulfonyl]-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.0027
N-[(4'-[1-[3-(trifluoromethyl)phenyl]ethoxy]biphenyl-4-yl)sulfonyl]-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.000086
N-[(4'-[[(3-methyl-1-benzofuran-2-yl)carbonyl]oxy]biphenyl-4-yl)sulfonyl]-D-valine
Rattus norvegicus
-
IC50: 0.000086 mM
0.0007
N-[(4'-[[(3-methyl-1-benzofuran-2-yl)oxy]methyl]biphenyl-4-yl)sulfonyl]-D-valine
Rattus norvegicus
-
IC50: 0.0007 mM
0.0091
N-[(4'-[[2-(trifluoromethyl)benzyl]oxy]biphenyl-4-yl)sulfonyl]-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.0022
N-[(4'-[[2-(trifluoromethyl)pyridin-4-yl]methoxy]biphenyl-4-yl)sulfonyl]-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.00076
N-[(4'-[[3-(methoxycarbonyl)benzyl]oxy]biphenyl-4-yl)sulfonyl]-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.00031
N-[(4'-[[3-(trifluoromethyl)benzyl]oxy]biphenyl-4-yl)sulfonyl]-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.0019
N-[(4'-[[4-(trifluoromethyl)benzyl]oxy]biphenyl-4-yl)sulfonyl]-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.0047
N-[(4'-[[6-(trifluoromethyl)pyridin-2-yl]methoxy]biphenyl-4-yl)sulfonyl]-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.2
N-[(4'-[[acetyl(methyl)amino]methyl]biphenyl-4-yl)sulfonyl]-D-valine
Homo sapiens
-
IC50 above 0.2 mM, pH and temperature not specified in the publication
0.000004
N-[[(4S)-4-(1-methylimidazol-2-yl)-2,5-dioxo-imidazolidin-4-yl]methyl]-5-(trifluoromethyl)benzofuran-2-carboxamide
Homo sapiens
pH 7.5, 22°C
0.0014
N-[[4'-(1-benzofuran-2-ylmethoxy)biphenyl-4-yl]sulfonyl]-D-valine
Rattus norvegicus
-
IC50: 0.0014 mM
0.0055
N-[[4'-(benzyloxy)biphenyl-4-yl]sulfonyl]-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.075
N-[[4'-(cyclohexylmethoxy)biphenyl-4-yl]sulfonyl]-D-valine
Homo sapiens
-
IC50 above 0.075 mM, pH and temperature not specified in the publication
0.0014
N-[[4'-(naphthalen-1-ylmethoxy)biphenyl-4-yl]sulfonyl]-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.0008
N-[[4'-(naphthalen-2-ylmethoxy)biphenyl-4-yl]sulfonyl]-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.033
N-[[4'-(pyridin-2-ylmethoxy)biphenyl-4-yl]sulfonyl]-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.03
N-[[4'-(pyridin-3-ylmethoxy)biphenyl-4-yl]sulfonyl]-D-valine
Homo sapiens
-
IC50 around 0.03 mM, pH and temperature not specified in the publication
0.0085
N-[[4'-(pyridin-4-ylmethoxy)biphenyl-4-yl]sulfonyl]-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.0106
N-[[4'-(quinolin-2-ylmethoxy)biphenyl-4-yl]sulfonyl]-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.001
N-[[4'-(quinolin-4-ylmethoxy)biphenyl-4-yl]sulfonyl]-D-valine
Homo sapiens
-
pH and temperature not specified in the publication
0.00021
N2-(biphenyl-4-ylcarbonyl)-N-(2-phenylpropan-2-yl)-L-alpha-glutamine
Homo sapiens
-
37°C, pH and temperature not specified in the publication
0.005
pyrogallol
Sus scrofa
-
pH 7.5, 37°C
0.000076
SE206
Bos taurus
-
macrocyclic derivate of BB-16, IC50: 76 nM