EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
4.6.1.18 | 0.00077 |
- |
ribonuclease inhibitor |
PE3I2 variant, pH 5.5, 25ºC |
654739 |
4.6.1.18 | 0.00078 |
- |
ribonuclease inhibitor |
C65A/C72A/G88R mutant, pH 6.0, 25ºC |
655979 |
4.6.1.18 | 0.0008 |
- |
ribonuclease inhibitor |
PE3I1 variant, pH 5.5, 25ºC |
654739 |
4.6.1.18 | 0.00134 |
- |
ribonuclease inhibitor |
PI5 variant, pH 5.5, 25ºC |
654739 |
4.6.1.18 | 0.0039 |
- |
ribonuclease inhibitor |
A4C/C65A/C72A/G88R/V118C mutant, pH 6.0, 25ºC |
655979 |
4.6.1.18 | 0.037 |
- |
3-amino-N-[2-hydroxymethyl-5-(5-methyl-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-tetrahydro-furan-3-yl]-succinamic acid |
pH 7.5, 25°C |
717371 |
4.6.1.18 | 0.067 |
- |
5'-carboxyadenosine |
pH 7.5, 25°C |
717371 |
4.6.1.18 | 0.075 |
- |
5'-deoxy-5'-N-(4-carboxypiperidinyl)uridine |
pH 7.5, 25°C |
717377 |
4.6.1.18 | 0.077 |
- |
1-(5-deoxy-5-[4-(ethoxycarbonyl)piperidin-1-yl]-alpha-L-arabinofuranosyl)pyrimidine-2,4(1H,3H)-dione |
- |
709463 |
4.6.1.18 | 0.08 |
- |
2',3'-dideoxy-3'-L-serinylamino thymidine |
- |
707728 |