EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
    6.2.1.3 | 0.0001 |
- |
Triacsin C |
inhibition of triacylglycerol synthesis |
692792 |
| 6.2.1.3 | 0.00016 |
- |
Triacsin A |
inhibition of triacylglycerol synthesis |
692792 |
| 6.2.1.3 | 0.00018 |
- |
Triacsin A |
inhibition of cholesteryl ester synthesis |
692792 |
| 6.2.1.3 | 0.00019 |
- |
Triacsin C |
inhibition of cholesteryl ester synthesis |
692792 |
| 6.2.1.3 | 0.0005 |
- |
rosiglitazone |
IC50: 0.0005 mM for ACS1-Flag fusion protein, no effect on ACS4-Flag fusion protein and ACS5-Flag fusion protein |
652138 |
| 6.2.1.3 | 0.0015 |
- |
pioglitazone |
IC50: 0.0015 mM for ACS1-Flag fusion protein, no effect on ACS4-Flag fusion protein and ACS5-Flag fusion protein |
652138 |
| 6.2.1.3 | 0.0015 |
- |
troglitazone |
IC50: 0.0015 mM for ACS1-Flag fusion protein, no effect on ACS4-Flag fusion protein and ACS5-Flag fusion protein |
652138 |
| 6.2.1.3 | 0.0055 |
- |
Triacsin C |
IC50: 0.0055 mM |
661181 |
| 6.2.1.3 | 0.0057 |
- |
5'-deoxy-5'-[([(1E)-5-[2-(methoxycarbonyl)phenyl]-5-oxopent-1-en-1-yl]sulfonyl)amino]adenosine |
- |
691308 |
| 6.2.1.3 | 0.02 |
- |
troglitazone |
no effect on FATP4 acyl-CoA synthetase activity towards n-tetracosanoic acid up to 0.05 mM, inhibits activity with palmitate with IC50 of 0.02 mM |
662341 |
