EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
7.6.2.2 | -999 |
- |
more |
data for drug inhibition of the basal ATPase activity |
659295 |
7.6.2.2 | -999 |
- |
more |
inhibition kinetics, overview |
697202 |
7.6.2.2 | 0.00028 |
0.00034 |
1,13-bis[4'-(4H-chromen-4-on-2-yl)phenyl]-N-(benzyl)-1,4,10,13-tetraoxa-7-azatridecane |
at 37°C, pH not specified in the publication |
734441 |
7.6.2.2 | 0.00042 |
- |
(2aR,6aS,12bR,14bS)-10,17-dimethoxy-3,3,6,6-tetramethyl-2a,3,6a,7,12b,14b-hexahydro-2H,6H-chromeno[3,4-c]chromeno[4',3':4,5]pyrano[3,2-h]chromene-13,14-dione |
recombinant MDR1in NIH-3T3 cells |
699450 |
7.6.2.2 | 0.00051 |
- |
(6aS,9bR,15aS,18bR)-3,12-dimethoxy-7,7,16,16-tetramethyl-6a,15a,16,18b-tetrahydro-6H,15H-chromeno[3,4-c]chromeno[4',3':4,5]pyrano[2,3-g]chromene-9,18(7H,9bH)-dione |
recombinant MDR1in NIH-3T3 cells |
699450 |
7.6.2.2 | 0.0006 |
- |
Hoechst 33342 |
at pH 7.5 and 37°C |
734258 |
7.6.2.2 | 0.00077 |
- |
(2R,4aR,7bR,9R,11aR,14bR)-2,5,5,9,12,12-hexamethyl-1,3,4,4a,5,8,9,10,11,11a,12,14b-dodecahydrobenzo[c]isochromeno[3,4-g]chromene-7,14(2H,7bH)-dione |
recombinant MDR1in NIH-3T3 cells |
699450 |
7.6.2.2 | 0.001 |
- |
(2aR,6aR,12bS,14bS)-10,17-dimethoxy-3,3,6,6-tetramethyl-2a,3,6a,7,12b,14b-hexahydro-2H,6H-chromeno[3,4-c]chromeno[4',3':4,5]pyrano[3,2-h]chromene-13,14-dione |
recombinant MDR1in NIH-3T3 cells |
699450 |
7.6.2.2 | 0.001 |
- |
(6aS,9bR,15aS,18bR)-2,4,11,13-tetrabromo-7,7,16,16-tetramethyl-6a,15a,16,18b-tetrahydro-6H,15H-chromeno[3,4-c]chromeno[4',3':4,5]pyrano[2,3-g]chromene-9,18(7H,9bH)-dione |
recombinant MDR1in NIH-3T3 cells |
699450 |
7.6.2.2 | 0.002 |
- |
cyclosporine A |
pH and temperature not specified in the publication |
733539 |