EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.1.3.48 | 0.00001 |
- |
ISIS 113715 |
IC50 less than 0.00001 mM |
692092 |
3.1.3.48 | 0.00015 |
- |
3-(4-carboxy-benzyloxy)-28-[4-butyric((s)-1-carboxyphenylethyl)-amide]-DELTA12-oleanene |
- |
691239 |
3.1.3.48 | 0.00017 |
- |
(2R)-2-benzyl-3-[2,6-dibromo-4-(6-bromo-5a,11a-dihydrobenzo[b]naphtho[2,3-d]furan-11-yl)phenyl]propanoic acid |
- |
679229 |
3.1.3.48 | 0.00019 |
- |
aquastatin A |
- |
707683 |
3.1.3.48 | 0.00021 |
- |
6-chloro-7-[(2-morpholin-4-ylethyl)amino]quinoline-5,8-dione |
- |
679229 |
3.1.3.48 | 0.00022 |
- |
4-[(2,4-dihydroxy-6-pentadecylbenzoyl)oxy]-2-hydroxy-6-methylbenzoic acid |
- |
707683 |
3.1.3.48 | 0.0003 |
- |
6-chloro-7-(2,3-dihydro-1H-inden-1-ylamino)quinoline-5,8-dione |
- |
679229 |
3.1.3.48 | 0.0003 |
- |
NSC-87877 |
Shp2, in 25 mM MOPS (pH 7.0), 50 mM NaCl, 0.05% (v/v) Tween 20, 1 mM dithiothreitol, at 25°C |
693564 |
3.1.3.48 | 0.00037 |
- |
methyl 5-amino-6-(7-amino-6-methoxy-5,8-dioxo-5,8-dihydroquinolin-2-yl)-4-(2-hydroxy-3,4-dimethoxyphenyl)-3-methylpyridine-2-carboxylate |
- |
679229 |
3.1.3.48 | 0.00038 |
- |
(2E)-2-[[5-(3-carboxy-4-hydroxycyclohexa-1,5-dien-1-yl)furan-2-yl]methylidene]-1-[6-[(4-fluorophenyl)amino][1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]diazanide |
pH and temperature not specified in the publication |
729370 |