EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   2.8.2.15 | 0.0016 |
- |
adenosine 3',5'-bisphosphate |
pH 7.5 |
645729 |
| 2.8.2.15 | 0.0028 |
- |
endoxifen |
with dehydroepiandrosterone as substrate, at pH 7.4 and 37°C |
738099 |
| 2.8.2.15 | 0.0035 |
- |
endoxifen |
with pregnenolone as substrate, at pH 7.4 and 37°C |
738099 |
| 2.8.2.15 | 0.0038 |
- |
androsterone |
pH 7.5, 37°C |
662232 |
| 2.8.2.15 | 0.008 |
- |
dehydroepiandrosterone |
in 0.25 M potassium phosphate buffer (pH 7.0), at 37°C |
724113 |
| 2.8.2.15 | 0.0096 |
- |
tamoxifen N-oxide |
with dehydroepiandrosterone as substrate, at pH 7.4 and 37°C |
738099 |
| 2.8.2.15 | 0.0098 |
- |
N-demethyltamoxifen |
with pregnenolone as substrate, at pH 7.4 and 37°C |
738099 |
| 2.8.2.15 | 0.0106 |
- |
dehydroepiandrosterone |
pH 7.5, 37°C |
662232 |
| 2.8.2.15 | 0.0127 |
- |
4-hydroxytamoxifen |
with pregnenolone as substrate, at pH 7.4 and 37°C |
738099 |
| 2.8.2.15 | 0.0169 |
- |
tamoxifen N-oxide |
with pregnenolone as substrate, at pH 7.4 and 37°C |
738099 |
