3.4.21.10: acrosin

This is an abbreviated version!
For detailed information about acrosin, go to the full flat file.

Word Map on EC 3.4.21.10

3.4.21.10

spermatozoa

semen

boar

pellucida

ejaculate

seminal

infertility

capacitation

oocyte

epididymal

trypsin-like

gamete

bull

contraceptive

ram

spermatid

zymogen

spermatogenesis

hyaluronidase

cryopreserved

benzamidine

antifertility

autoactivation

cauda

sperm-zona

kallikreins

acrosome-reacted

gelatinolytic

insemination

sperm-associated

asthenozoospermia

andrology

sperm-oocyte

nonoxynol-9

acrosome-intact

sperm-egg

p-aminobenzamidine

zona-free

analysis

spermatogonial

bapna

medicine

tlck

kazal-type

Reaction

preferential cleavage: Arg-/-, Lys-/- =

Synonyms

53 kDa fucose-binding protein, acrosin, acrosin amidase, acrosin I, acrosin II, acrosomal protease, acrosomal proteinase, acrozonase, alpha-acrosin, beta-acrosin, proteinase, acrosomal, psi-acrosin, sperm acrosin

ECTree

3 Hydrolases

3.4 Acting on peptide bonds (peptidases)

3.4.21 Serine endopeptidases

3.4.21.10 acrosin

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Results	in table
5	Activating Compound
167	AA Sequence
7	Application
1	CAS Registry Number
1	Cloned(Commentary)
2	Crystallization (Commentary)
318	Disease/ Diagnostics
2	Expression
4	General Information
10	General Stability
160	IC50 Value
285	Inhibitors
1	Ki Value [mM]
15	KM Value [mM]
10	Localization
7	Metals/Ions
69	Molecular Weight [Da]
170	Natural Substrates/ Products (Substrates)
115	Organism
15	pH Optimum
3	pH Range
5	pH Stability
2	pI Value
9	Posttranslational Modification
1	Protein Variants
19	Purification (Commentary)
1	Reaction
1	Reaction Type
114	Reference
102	Source Tissue
12	Specific Activity [micromol/min/mg]
4	Storage Stability
202	Substrates and Products (Substrate)
69	Subunits
61	Synonyms
3	Temperature Optimum [°C]
1	Temperature Range [°C]
1	Temperature Stability [°C]
5	Turnover Number [1/s]

IC50 Value

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IC50 Value on EC 3.4.21.10 - acrosin

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3.78

1-(2,4-dichlorobenzoyl)-N-methyl-1H-indazole-3-carboxamide

Homo sapiens

pH and temperature not specified in the publication

731747

0.00563

2,4-dichloro-N-[4-[(diaminomethylidene)sulfamoyl]phenyl]benzamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00596

2,6-dichloro-N-[4-[(diaminomethylidene)sulfamoyl]phenyl]benzamide

Homo sapiens

pH and temperature not specified in the publication

717359

6.04

2-(3-(2-hydroxyethyl)ureido)-N-(2-methoxybenzyl)-1H-benzo[d]imidazole-5-sulfonamide

Homo sapiens

pH and temperature not specified in the publication

731747

5.45

2-(3-(2-hydroxyethyl)ureido)-N-(2-methylbenzyl)-1H-benzo[d]imidazole-5-sulfonamide

Homo sapiens

pH and temperature not specified in the publication

731747

0.00935

2-(4-chlorophenoxy)-N-[4-[(diaminomethylidene)sulfamoyl]phenyl]acetamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00763

2-bromo-N-[4-[(diaminomethylidene)sulfamoyl]phenyl]benzamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.0063

2-chloro-N-[4-[(diaminomethylidene)sulfamoyl]phenyl]benzamide

Homo sapiens

pH and temperature not specified in the publication

717359

7.32

2-{[(2-hydroxyethyl)carbamoyl]amino}-N-[(2-methoxyphenyl)methyl]-1H-benzimidazole-5-sulfonamide

Homo sapiens

pH and temperature not specified in the publication

731747

0.0038

3,4-dichloro-N-[4-[(diaminomethylidene)sulfamoyl]phenyl]benzamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.42

3-(4-nitrophenyl)-1,2-oxazole-5-carbaldehyde

Homo sapiens

in 55 mM HEPES and 55 mM NaCl at pH 8.0 and 37°C

717912

0.007

3-chloro-N-[4-[(diaminomethylidene)sulfamoyl]phenyl]benzamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00251

3-methylbutyl 1-[2-([4-[(diaminomethylidene)sulfamoyl]phenyl]amino)-2-oxoethyl]piperidine-4-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717359

0.0033

3-[4-([[4-(aminomethyl)cyclohexyl]carbonyl]oxy)phenyl]propanoic acid

Homo sapiens

in 55 mM HEPES and 55 mM NaCl at pH 8.0 and 37°C

717912

0.008

4-(acetylamino)phenyl 4-carbamimidamidobenzoate

Homo sapiens

in 55 mM HEPES and 55 mM NaCl at pH 8.0 and 37°C

717912

0.00384

4-(chloromethyl)-N-[4-[(diaminomethylidene)sulfamoyl]phenyl]benzamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00925

4-([4-[3-(ethoxycarbonyl)-1H-pyrazol-5-yl]phenyl]amino)-4-oxobutanoic acid

Homo sapiens

pH and temperature not specified in the publication

717353

0.3447

4-[(2-methylbenzyl)(methylsulfonyl)amino]-N-(pyridin-4-ylmethyl)benzamide

Homo sapiens

in 55 mM HEPES and 55 mM NaCl at pH 8.0 and 37°C

717912

0.39 - 1.7

5-(2,4-dichlorophenyl)-1,2-oxazole-3-carbaldehyde

3 entries

0.1

5-(4-carbamimidamidophenyl)-N-(1-hydroxypropan-2-yl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0115

5-(4-carbamimidamidophenyl)-N-(2,3-dimethylphenyl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0014

5-(4-carbamimidamidophenyl)-N-(2,4-dimethoxyphenyl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0023

5-(4-carbamimidamidophenyl)-N-(2,5-dimethoxyphenyl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0057

5-(4-carbamimidamidophenyl)-N-(2,6-dimethylphenyl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0084

5-(4-carbamimidamidophenyl)-N-(2-methoxyphenyl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0144

5-(4-carbamimidamidophenyl)-N-(2-methylphenyl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0121

5-(4-carbamimidamidophenyl)-N-(3,5-dimethylphenyl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0254

5-(4-carbamimidamidophenyl)-N-(3-chlorophenyl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0066

5-(4-carbamimidamidophenyl)-N-(3-methoxyphenyl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0094

5-(4-carbamimidamidophenyl)-N-(3-methylphenyl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0268

5-(4-carbamimidamidophenyl)-N-(4-chlorophenyl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0239

5-(4-carbamimidamidophenyl)-N-(4-cyanophenyl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0064

5-(4-carbamimidamidophenyl)-N-(4-ethoxyphenyl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0205

5-(4-carbamimidamidophenyl)-N-(4-fluorophenyl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0101

5-(4-carbamimidamidophenyl)-N-(4-methylphenyl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0214

5-(4-carbamimidamidophenyl)-N-(4-methylpyridin-2-yl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0299

5-(4-carbamimidamidophenyl)-N-(naphthalen-1-yl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.1

5-(4-carbamimidamidophenyl)-N-(propan-2-yl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0246

5-(4-carbamimidamidophenyl)-N-phenyl-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

0.0203

5-(4-carbamimidamidophenyl)-N-[4-(trifluoromethyl)phenyl]-1,2-oxazole-3-carboxamide hydrochloride

Homo sapiens

pH 7.8, 37.8°C

731451

0.0174

5-([4-[3-(ethoxycarbonyl)-1H-pyrazol-5-yl]phenyl]amino)-5-oxopentanoic acid

Homo sapiens

pH and temperature not specified in the publication

717353

0.0095

butyl 1-[2-([4-[(diaminomethylidene)sulfamoyl]phenyl]amino)-2-oxoethyl]piperidine-4-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717359

3.24

ethyl 1-(2,4-dichlorobenzoyl)-1H-indazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

731747

0.00221

ethyl 1-(phenylcarbonyl)-1H-pyrrolo[2,3-b]pyridine-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717498

0.00029

ethyl 1-[(2,4-dichlorophenyl)carbonyl]-1H-pyrrolo[2,3-b]pyridine-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717498

0.00174

ethyl 1-[(2-bromo-4-fluorophenyl)carbonyl]-1H-pyrrolo[2,3-b]pyridine-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717498

0.00347

ethyl 1-[(2-chloro-4-fluorophenyl)carbonyl]-1H-pyrrolo[2,3-b]pyridine-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717498

0.00299

ethyl 1-[2-([4-[(diaminomethylidene)sulfamoyl]phenyl]amino)-2-oxoethyl]piperidine-4-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717359

0.0093

ethyl 4-([[5-(4-carbamimidamidophenyl)-1,2-oxazol-3-yl]carbonyl]amino)benzoate hydrochloride

Homo sapiens

pH 7.8, 37.8°C

731451

0.00044

ethyl 5-(4-[[(2,4-dichlorophenyl)carbonyl]amino]phenyl)-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.0048

ethyl 5-(4-[[(2,6-dichlorophenyl)carbonyl]amino]phenyl)-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.00398

ethyl 5-(4-[[(2,6-difluorophenyl)carbonyl]amino]phenyl)-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.0024

ethyl 5-(4-[[(2-bromophenyl)carbonyl]amino]phenyl)-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.00011

ethyl 5-(4-[[(2-chlorophenyl)carbonyl]amino]phenyl)-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.00331

ethyl 5-(4-[[(4-chlorophenyl)carbonyl]amino]phenyl)-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.0024

ethyl 5-(4-[[(4-fluorophenyl)carbonyl]amino]phenyl)-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.0008

ethyl 5-(4-[[(4-methoxyphenyl)carbonyl]amino]phenyl)-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.0346

ethyl 5-(4-[[(4-methylphenyl)carbonyl]amino]phenyl)-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.0033

ethyl 5-(4-[[4-(1-phenylpropyl)benzoyl]amino]phenyl)-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.023

ethyl 5-[4-(acetylamino)phenyl]-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.46

ethyl 5-[4-(benzoylamino)phenyl]-1,2-oxazole-3-carboxylate

Homo sapiens

pH 7.8, 37.8°C

731451

0.017

ethyl 5-[4-(butanoylamino)phenyl]-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.072

ethyl 5-[4-(pentanoylamino)phenyl]-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.014

ethyl 5-[4-(propanoylamino)phenyl]-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.000032

ethyl 5-[4-([4-[(4-methylphenyl)sulfonyl]benzoyl]amino)phenyl]-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.00331

ethyl 5-[4-([[4-(chloromethyl)phenyl]carbonyl]amino)phenyl]-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.06

ethyl 5-[4-[(2-chlorobenzoyl)amino]phenyl]-1,2-oxazole-3-carboxylate

Homo sapiens

pH 7.8, 37.8°C

731451

0.24

ethyl 5-[4-[(3,4-dichlorobenzoyl)amino]phenyl]-1,2-oxazole-3-carboxylate

Homo sapiens

pH 7.8, 37.8°C

731451

0.00576

ethyl 5-[4-[(3-chloropropanoyl)amino]phenyl]-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.00047

ethyl 5-[4-[(4-benzylbenzoyl)amino]phenyl]-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.38

ethyl 5-[4-[(4-chlorobenzoyl)amino]phenyl]1,2-oxazole-3-carboxylate

Homo sapiens

pH 7.8, 37.8°C

731451

0.14

ethyl 5-[4-[(4-fluorobenzoyl)amino]phenyl]-1,2-oxazole-3-carboxylate

Homo sapiens

pH 7.8, 37.8°C

731451

0.008

ethyl 5-[4-[(phenylcarbonyl)amino]phenyl]-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.0079

ethyl 5-[4-[(trifluoroacetyl)amino]phenyl]-1H-pyrazole-3-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717353

0.000027

KF950

Homo sapiens

pH and temperature not specified in the publication

717359

10.7

methyl (6-[[4-(trifluoromethyl)phenyl]sulfamoyl]-1H-benzimidazol-2-yl)carbamate

Homo sapiens

pH 8.0, 22°C

731432

0.0093

methyl 1-[2-([4-[(diaminomethylidene)sulfamoyl]phenyl]amino)-2-oxoethyl]piperidine-4-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717359

0.1555

methyl 4-methyl-3-([4-[(2-methylbenzyl)(methylsulfonyl)amino]benzoyl]amino)benzoate

Homo sapiens

in 55 mM HEPES and 55 mM NaCl at pH 8.0 and 37°C

717912

1.77

methyl [6-(butylsulfamoyl)-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

1.8

methyl [6-(hexylsulfamoyl)-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

1.03

methyl [6-(phenylsulfamoyl)-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

0.47

methyl [6-(propan-2-ylsulfamoyl)-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

1.27

methyl [6-[(2,4-dichlorophenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

1.55

methyl [6-[(2,4-difluorophenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

8.86

methyl [6-[(2,5-dimethylphenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

5.75

methyl [6-[(2-chlorophenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

0.31

methyl [6-[(2-fluorophenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

8.42

methyl [6-[(2-methoxyphenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

4.02

methyl [6-[(3,4-dichlorophenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

1.59

methyl [6-[(3,4-difluorophenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

11.5

methyl [6-[(3,4-dimethoxyphenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

1.81

methyl [6-[(3-fluorophenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

7.5

methyl [6-[(3-methoxyphenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

5.06

methyl [6-[(3-methylphenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

1.64

methyl [6-[(4-bromophenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

7.52

methyl [6-[(4-chlorophenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

2.4

methyl [6-[(4-fluorophenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

3.29

methyl [6-[(4-methoxyphenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

3.18

methyl [6-[(4-methylphenyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

1.25

methyl [6-[benzyl(methyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

0.063

methyl [6-[bis(3-methylbutyl)sulfamoyl]-1H-benzimidazol-2-yl]carbamate

Homo sapiens

pH 8.0, 22°C

731432

5.73

N,N-bis(2-hydroxyethyl)-5-(4-methoxyphenyl)-1H-pyrazole-3-carboxamide

Homo sapiens

pH and temperature not specified in the publication

731747

0.4267

N,N-dibenzyl-2-[4-(propan-2-ylsulfamoyl)phenoxy]acetamide

Homo sapiens

in 55 mM HEPES and 55 mM NaCl at pH 8.0 and 37°C

717912

0.0279

N-(2-bromophenyl)-5-(4-carbamimidamidophenyl)-1,2-oxazole-3-carboxamide

Homo sapiens

pH 7.8, 37.8°C

731451

1.06

N-(2-chlorobenzyl)-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide

Homo sapiens

pH and temperature not specified in the publication

731747

0.08

N-(2-fluorobenzyl)-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide

Homo sapiens

pH and temperature not specified in the publication

731747

6.81

N-(2-hydroxyethyl)-5-(4-methoxyphenyl)-N-methyl-1H-pyrazole-3-carboxamide

Homo sapiens

pH and temperature not specified in the publication

731747

8.92

N-(2-hydroxypropyl)-5-(4-methoxyphenyl)-1H-pyrazole-3-carboxamide

Homo sapiens

pH and temperature not specified in the publication

731747

0.34

N-(3, 5-difluorobenzyl)-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide

Homo sapiens

pH and temperature not specified in the publication

731747

2.45

N-(3,5-dichlorobenzyl)-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide

Homo sapiens

pH and temperature not specified in the publication

731747

0.0144

N-(3-bromophenyl)-5-(4-carbamimidamidophenyl)-1,2-oxazole-3-carboxamide hydrochloride

Homo sapiens

pH 7.8, 37.8°C

731451

1.43

N-(3-hydroxypropyl)-5-(4-methoxyphenyl)-1H-pyrazole-3-carboxamide

Homo sapiens

pH and temperature not specified in the publication

731747

0.014

N-(4-chlorophenyl)-N-[2-[(2E)-2-(3-methoxy-4-methylbenzylidene)hydrazinyl]-2-oxoethyl]benzenesulfonamide (non-preferred name)

Homo sapiens

in 55 mM HEPES and 55 mM NaCl at pH 8.0 and 37°C

717912

0.0078

N-(4-tert-butylphenyl)-5-(4-carbamimidamidophenyl)-1,2-oxazole-3-carboxamide hydrochloride

Homo sapiens

pH 7.8, 37.8°C

731451

5.08

N-(5-bromobenzo[d]thiazol-2-yl)-2-(4-pentylpiperazin-1-yl)acetamide

Homo sapiens

pH and temperature not specified in the publication

731747

1.09

N-(5-bromobenzo[d]thiazol-2-yl)-2-(diisopentylamino)acetamide

Homo sapiens

pH and temperature not specified in the publication

731747

0.54

N-(5-bromobenzo[d]thiazol-2-yl)-2-(dipentylamino)acetamide

Homo sapiens

pH and temperature not specified in the publication

731747

2.78

N-(6-bromobenzo[d]thiazol-2-yl)-2-(dibutylamino)acetamide

Homo sapiens

pH and temperature not specified in the publication

731747

142.6

N-alpha-tosyl-L-lysyl-chloromethyl-ketone

Homo sapiens

pH and temperature not specified in the publication

731747

0.1426

N-alpha-tosyl-L-lysyl-chloromethylketone

2 entries

0.28

N-benzyl-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide

Homo sapiens

pH and temperature not specified in the publication

731747

0.3551

N-cyclohexyl-2-[(4,6-diphenylpyrimidin-2-yl)sulfanyl]acetamide

Homo sapiens

in 55 mM HEPES and 55 mM NaCl at pH 8.0 and 37°C

717912

1.62

N-hexyl-2-(3-(2-hydroxyethyl)ureido)-1H-benzo[d]imidazole-5-sulfonamide

Homo sapiens

pH and temperature not specified in the publication

731747

0.1426

N-tosyl-L-lysine chloromethylketone

Homo sapiens

pH and temperature not specified in the publication

717498

0.3018

N-[4-(dipropylsulfamoyl)phenyl]-3,4-diethoxybenzamide

Homo sapiens

in 55 mM HEPES and 55 mM NaCl at pH 8.0 and 37°C

717912

0.6248

N-[4-[(4-benzylpiperazin-1-yl)carbonyl]phenyl]-2,3,5,6-tetramethylbenzenesulfonamide

Homo sapiens

in 55 mM HEPES and 55 mM NaCl at pH 8.0 and 37°C

717912

3.057

N-[4-[(4-benzylpiperazin-1-yl)carbonyl]phenyl]-4-tert-butylbenzenesulfonamide

Homo sapiens

in 55 mM HEPES and 55 mM NaCl at pH 8.0 and 37°C

717912

0.2053

N-[4-[(4-fluorophenyl)sulfamoyl]phenyl]-3,4,5-trimethoxybenzamide

Homo sapiens

in 55 mM HEPES and 55 mM NaCl at pH 8.0 and 37°C

717912

0.6678

N-[4-[(4-methoxyphenyl)sulfamoyl]phenyl]-2-(naphthalen-1-yloxy)acetamide

Homo sapiens

in 55 mM HEPES and 55 mM NaCl at pH 8.0 and 37°C

717912

0.00245

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-2,4,6-trimethylbenzamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00718

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-2,6-difluorobenzamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.0093

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-2-(2-methylphenoxy)acetamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.0099

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-2-(2-methylpiperidin-1-yl)acetamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00892

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-2-(3-methylphenoxy)acetamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00984

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-2-(4-methoxyphenoxy)acetamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00898

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-2-(4-methylphenoxy)acetamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00498

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-2-(4-methylpiperidin-1-yl)acetamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.0042

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-2-(4-nitrophenoxy)acetamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00741

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-2-(piperidin-1-yl)acetamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.0023

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-2-phenoxyacetamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.0025

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-3,5-dinitrobenzamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00705

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-3-(trifluoromethyl)benzamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00013

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-4-ethoxybenzamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00021

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-4-ethylbenzamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00711

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-4-fluorobenzamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00221

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-4-methoxybenzamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00206

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]-4-methylbenzamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00958

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]butanamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.00158

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]pentanamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.009

N-[4-[(diaminomethylidene)sulfamoyl]phenyl]propanamide

Homo sapiens

pH and temperature not specified in the publication

717359

0.012

NF064

Sus scrofa

23°C

679420

0.7

NSC651015

Sus scrofa

23°C

679420

0.7

NSC651016

Sus scrofa

23°C

679420

0.00235

propan-2-yl 1-[2-([4-[(diaminomethylidene)sulfamoyl]phenyl]amino)-2-oxoethyl]piperidine-4-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717359

0.00331

propyl 1-[2-([4-[(diaminomethylidene)sulfamoyl]phenyl]amino)-2-oxoethyl]piperidine-4-carboxylate

Homo sapiens

pH and temperature not specified in the publication

717359

0.1

suramin

Sus scrofa

23°C

679420