EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.25.1 | 0.000757 |
- |
syringolin A methyl ester |
for the chymotrypsin-like activity, pH not specified in the publication, temperature not specified in the publication |
713407 |
3.4.25.1 | 0.00084 |
- |
N-(tert-butoxycarbonyl)-L-alanyl-N5-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N1-(naphthalen-2-ylmethyl)-L-glutamamide |
chymotrypsin-like, b5 activity of 20S proteasome, pH not specified in the publication, temperature not specified in the publication |
707667 |
3.4.25.1 | 0.00102 |
- |
syringolin A |
for the chymotrypsin-like activity, pH not specified in the publication, temperature not specified in the publication |
713407 |
3.4.25.1 | 0.00147 |
- |
N-(tert-butoxycarbonyl)-L-phenylalanyl-N5-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N1-(naphthalen-2-ylmethyl)-L-glutamamide |
chymotrypsin-like, b5 activity of 20S proteasome, pH not specified in the publication, temperature not specified in the publication |
707667 |
3.4.25.1 | 0.0015 |
- |
N-(tert-butoxycarbonyl)-L-isoleucyl-N5-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N1-(naphthalen-2-ylmethyl)-L-glutamamide |
chymotrypsin-like, b5 activity of 20S proteasome, pH not specified in the publication, temperature not specified in the publication |
707667 |
3.4.25.1 | 0.00164 |
- |
N-(tert-butoxycarbonyl)-O-methyl-L-tyrosyl-N-[(2S)-1-(furan-2-yl)-4-methyl-1-oxopentan-2-yl]-L-tyrosinamide |
in 10 mM HEPES (pH 7.6), at 37°C |
733663 |
3.4.25.1 | 0.002 |
- |
glidobactin A |
for the trypsin-like activity, pH not specified in the publication, temperature not specified in the publication |
713407 |
3.4.25.1 | 0.00262 |
- |
N-[(benzyloxy)carbonyl]-L-phenylalanyl-N-[(2S)-1-(furan-2-yl)-4-methyl-1-oxopentan-2-yl]-O-methyl-L-tyrosinamide |
in 10 mM HEPES (pH 7.6), at 37°C |
733663 |
3.4.25.1 | 0.00274 |
- |
N-(tert-butoxycarbonyl)glycyl-N6-[(1R)-1-(dihydroxyboranyl)-3-methylbutyl]-N-(naphthalen-2-ylmethyl)-6-oxo-L-lysinamide |
chymotrypsin-like, b5 activity of 20S proteasome, pH not specified in the publication, temperature not specified in the publication |
707667 |
3.4.25.1 | 0.00327 |
- |
Nalpha-[(2S)-2-[[(benzyloxy)carbonyl]amino]-4-(4-methoxyphenyl)butanoyl]-N-[(2S)-1-(furan-2-yl)-4-methyl-1-oxopentan-2-yl]-L-tyrosinamide |
in 10 mM HEPES (pH 7.6), at 37°C |
733663 |