EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.25.1 | 0.056 |
- |
Benzyloxycarbonyl-Leu-Leu-Arg |
IC50: 0.056 mM for chymotrypsin-like activity, 0.0014 mM for trypsin-like activity |
650902 |
3.4.25.1 | 0.065 |
- |
benzyloxycarbonyl-Leu-Thr-Arg |
IC50: 0.065 mM for chymotrypsin-like activity, 0.0021 mM for trypsin-like activity |
650902 |
3.4.25.1 | 0.077 |
- |
NPLLNVS |
IC50: 0.063 mM, inhibition of hydrolysis of Gly-Gly-Arg-7-amido-4-carbamoylcoumarin. IC50: 0.077 mM, inhibition of hydrolysis of succinyl-Leu-Leu-Val-Tyr-7-amido-4-methylcoumarin |
652378 |
3.4.25.1 | 0.1 |
- |
leupeptin |
IC50: 0.0015 mM, inhibition of hydrolysis of Gly-Gly-Arg-7-amido-4-methylcoumarin, most potent inhibitor for hydrolysis of Gly-Gly-Arg-7-amido-4-methylcoumarin. IC50: 0.1 mM, inhibition of hydrolysis of succinyl-Leu-Leu-Val-Tyr-7-amido-4-methylcoumarin |
652378 |
3.4.25.1 | 0.1078 |
- |
syringolin B |
for the trypsin-like activity, pH not specified in the publication, temperature not specified in the publication |
713407 |
3.4.25.1 | 0.11 |
- |
benzyloxycarbonyl-Leu-Gly-Arg |
IC50: 0.11 mM for chymotrypsin-like activity, 0.0066 mM for trypsin-like activity |
650902 |
3.4.25.1 | 0.85 |
- |
acetyl-Leu-Leu-Arg |
IC50: 0.85 mM for chymotrypsin-like activity, 0.0056 mM for trypsin-like activity |
650902 |