EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.22.51 | 0.05 |
- |
N'-[(E)-(2,6-dichlorophenyl)methylidene]-3,4,5-trimethoxybenzohydrazide |
pH 6.5, 22°C |
717894 |
3.4.22.51 | 0.055 |
- |
N'-[(E)-(4-bromophenyl)methylidene]-3,4,5-trimethoxybenzohydrazide |
pH 6.5, 22°C |
717894 |
3.4.22.51 | 0.078 |
- |
N-phenyl benzofuroxan-5-carboxaldehyde thiosemicarbazone |
- |
696729 |
3.4.22.51 | 1.41 |
- |
N-[4-methyl-3-(piperidin-1-ylsulfonyl)phenyl]-4-oxo-4-(3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)butanamide |
23°C, pH 6.5 |
753924 |
3.4.22.51 | 0.1 |
- |
N4-allyl benzofuroxan-5-carboxaldehyde thiosemicarbazone |
above 0.1 mM |
696729 |
3.4.22.51 | 0.000004 |
- |
Nalpha-[(2R,3E)-2-benzyl-4-(phenylsulfonyl)but-3-enoyl]-N-[(4-methylpiperazin-1-yl)carbonyl]-L-phenylalaninamide |
- |
696645 |
3.4.22.51 | 0.0001 |
- |
Nalpha-[(2R,3E)-2-benzyl-4-(phenylsulfonyl)but-3-enoyl]-N-[(4-methylpiperazin-1-yl)carbonyl]-L-phenylalaninamide |
- |
696645 |
3.4.22.51 | 0.0077 |
- |
nifurtimox |
- |
696760 |
3.4.22.51 | 0.0228 |
- |
nitrofurazone |
pH 6.5, 37°C |
717917 |