EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
4.6.1.2 | -999 |
- |
more |
inhibition kinetics |
692446 |
4.6.1.2 | 0.00005 |
- |
Ca2+ |
- |
667002 |
4.6.1.2 | 0.00005 |
- |
Ca2+ |
soluble guanylyl cyclase sGC |
667002 |
4.6.1.2 | 0.0002 |
- |
Ca2+ |
soluble guanylyl cyclase sGC |
667002 |
4.6.1.2 | 0.00071 |
- |
2',3'-O-(2,4,6-trinitrophenyl)-ATP |
in 10 mM MnCl2, 100 mM KCl, 25 mM HEPES/NaOH, pH 7.4, at 30°C |
709679 |
4.6.1.2 | 0.001 |
- |
Go6976 |
in the presence of 1 mM ATP, isozyme GC-A, in 25 mM HEPES (pH 7.4), 50 mM NaCl, 0.1% (w/v) bovine serum albumin, 0.5 mM isobutylmethyl xanthine, 1 mM EDTA, 0.5 mM microcystin and 5 mM MgCl2, at 37°C |
715634 |
4.6.1.2 | 0.0013 |
- |
Go6976 |
in the presence of 1 mM ATP, isozyme GC-B, in 25 mM HEPES (pH 7.4), 50 mM NaCl, 0.1% (w/v) bovine serum albumin, 0.5 mM isobutylmethyl xanthine, 1 mM EDTA, 0.5 mM microcystin and 5 mM MgCl2, at 37°C |
715634 |
4.6.1.2 | 0.00311 |
- |
2',3'-O-(2,4,6-trinitrophenyl)-UTP |
in 10 mM MnCl2, 100 mM KCl, 25 mM HEPES/NaOH, pH 7.4, at 30°C |
709679 |
4.6.1.2 | 0.0051 |
- |
2',3'-O-(2,4,6-trinitrophenyl)-CTP |
in 10 mM MnCl2, 100 mM KCl, 25 mM HEPES/NaOH, pH 7.4, at 30°C |
709679 |
4.6.1.2 | 0.0051 |
- |
AMP-PNP |
at 10°C |
680671 |