EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.1.1.45 | 0.000018 |
- |
(2R)-2-(5-[[(1-hydroxy-3-methyl-5,10a-dihydrobenzo[f]quinazolin-9-yl)methyl]amino]-1-oxo-1,3-dihydro-2H-isoindol-2-yl)butanedioic acid |
22°C |
694812 |
2.1.1.45 | 0.0027 |
- |
1,3-propanediphosphonic acid |
pH 7.2, 22°C |
690892 |
2.1.1.45 | 0.016 |
- |
1-(2'-deoxyribosyl)-8-azapurin-2-one 5'-monophosphate |
- |
485385 |
2.1.1.45 | 0.12 |
- |
1-(beta-D-2'-deoxyribofuranosyl)-1,6-dihydro-8-azapurin-2(3H,6H)-one 5'-monophosphate |
- |
485385 |
2.1.1.45 | 0.022 |
- |
1-(beta-D-2-deoxyribofuranosyl)-4-hydroxyamino-5-bromopyrimidin-2(1H)-one 5'-monophosphate |
L1210 recombinant enzyme |
485427 |
2.1.1.45 | 0.0321 |
- |
1-(beta-D-2-deoxyribofuranosyl)-4-hydroxyamino-5-bromopyrimidin-2(1H)-one 5'-monophosphate |
L1210 parental enzyme |
485427 |
2.1.1.45 | 0.0049 |
- |
1-(beta-D-2-deoxyribofuranosyl)-4-hydroxyamino-5-chloropyrimidin-2(1H)-one 5'-monophosphate |
L1210 recombinant enzyme |
485427 |
2.1.1.45 | 0.0085 |
- |
1-(beta-D-2-deoxyribofuranosyl)-4-hydroxyamino-5-chloropyrimidin-2(1H)-one 5'-monophosphate |
L1210 parental enzyme |
485427 |
2.1.1.45 | 0.0008 |
- |
1-(beta-D-2-deoxyribofuranosyl)-4-hydroxyamino-5-fluoropyrimidin-2(1H)-one 5'-monophosphate |
L1210 parental enzyme |
485427 |
2.1.1.45 | 0.0014 |
- |
1-(beta-D-2-deoxyribofuranosyl)-4-hydroxyamino-5-fluoropyrimidin-2(1H)-one 5'-monophosphate |
L1210 recombinant enzyme |
485427 |