EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
5.1.1.4 | 0.0036 |
- |
pyrrole-2-carboxylic acid |
pH 6.0, 37°C, TcPRACB |
652377 |
5.1.1.4 | 0.0057 |
- |
pyrrole-2-carboxylic acid |
pH 6.0, 37°C, TcPRACA |
652377 |
5.1.1.4 | 0.02 |
- |
pyrrole-2-carboxylic acid |
0.005 mM pyrrole-2-carboxylic acid, serial concentrations of 20-160 mM L-proline |
705596 |
5.1.1.4 | 111 |
- |
tetrahydro-1H-pyrrolizine-7a(5H)-carboxylate |
pH and temperature not specified in the publication |
727156 |
5.1.1.4 | 0.006 |
0.01 |
2-pyrrolecarboxylic acid |
recombinant His-tagged enzyme, pH 6.0, 37°C |
728600 |
5.1.1.4 | 0.3 |
- |
4-chloropyrazole-3-carboxylic acid |
recombinant His-tagged enzyme, pH 6.0, 37°C |
728600 |
5.1.1.4 | 1 |
- |
4-bromopyrazole-3-carboxylic acid |
recombinant His-tagged enzyme, pH 6.0, 37°C |
728600 |
5.1.1.4 | 2 |
- |
4-chloro-5-methyl-pyrazole-3-carboxylic acid |
recombinant His-tagged enzyme, pH 6.0, 37°C |
728600 |
5.1.1.4 | 2 |
- |
4-ethylpyrazole-3-carboxylic acid |
recombinant His-tagged enzyme, pH 6.0, 37°C |
728600 |
5.1.1.4 | 2 |
- |
pyrazole-3-carboxylic acid |
recombinant His-tagged enzyme, pH 6.0, 37°C |
728600 |