EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.5.4.4 | 0.029 |
- |
5'-methylthiocoformycin |
wild type enzyme, in 100 mM Tris-HCl buffer (pH 8.0), temperature not specified in the publication |
711215 |
3.5.4.4 | 0.0009 |
- |
(2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-2-ol |
mutant D172A, pH 7.5, 30°C |
718893 |
3.5.4.4 | 0.0019 |
- |
(2S,3R)-3-(6-amino-9H-purin-9-yl)nonan-2-ol |
wild-type, pH 7.5, 30°C |
718893 |
3.5.4.4 | 0.0005 |
- |
erythro-9-(2-hydroxy-3-nonyl)adenine |
pH 7.4, 37°C |
719423 |
3.5.4.4 | 0.00000025 |
- |
coformycin |
37°C, pH not specified in the publication |
720969 |
3.5.4.4 | 0.0000034 |
- |
2'-deoxycoformycin |
37°C, pH not specified in the publication |
720969 |
3.5.4.4 | 0.00000011 |
- |
(2S,3R)-3-(6-amino-9H-purin-9-yl)-5-[3-(trifluoromethyl)phenyl]pentan-2-ol |
pH 7.0, temperature not specified in the publication |
752963 |
3.5.4.4 | 0.0000022 |
- |
(+)-erythro-9-(2-hydroxy-3-nonyl)adenine |
pH 7.0, temperature not specified in the publication |
752963 |
3.5.4.4 | 0.0000052 |
- |
(2S,3R)-3-(6-amino-9H-purin-9-yl)-5-[4-(trifluoromethyl)phenyl]pentan-2-ol |
pH 7.0, temperature not specified in the publication |
752963 |
3.5.4.4 | 0.0000059 |
- |
1-[(3R,4S)-4-hydroxy-1-[3-(trifluoromethyl)phenyl]pentan-3-yl]-1H-imidazole-4-carboxamide |
pH 7.0, temperature not specified in the publication |
752963 |