EC Number   |
Inhibitors |
Structure |
|---|
    3.1.1.79 | 4-methoxyphenyl 3,4-dihydroisoquinolin-2(1H)-ylcarbamate |
IC50: 360 nM |
   |
| 3.1.1.79 | 4-[(2,2-dimethylpropanoyl)amino]phenyl morpholin-4-ylcarbamate |
IC50: 47 nM |
|
| 3.1.1.79 | 4-[(cyclohexylcarbonyl)amino]phenyl morpholin-4-ylcarbamate |
IC50: 10 nM |
|
| 3.1.1.79 | 76-0079 |
a commercial small molecule inhibitor |
|
| 3.1.1.79 | Ba2+ |
10 mM, 40% loss of activity |
|
| 3.1.1.79 | benzyl (4-(5-methoxy-2-oxo-1,3,4-oxadiazol-3(2H)-yl)-2-methylphenyl)carbamate |
- |
|
| 3.1.1.79 | benzyl (4-[[(morpholin-4-ylamino)carbonyl]oxy]phenyl)acetate |
IC50: 5 nM |
|
| 3.1.1.79 | betaine |
it enhances the enzyme activity 2fold at 50°C and 3 M, and 1.5fold at 45°C and 1-3 M, while it reduces the enzyme activity at 35-40°C, by 20% at 40°C and 3 M,about % at 1 M, overview |
|
| 3.1.1.79 | CaCl2 |
50 mM, 47% inhibition |
|
| 3.1.1.79 | CAY10499 |
- |
|
