EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
5.3.99.2 | 0.1 |
- |
1-benzoyl piperazine |
larger than 0.100 mM |
703559 |
5.3.99.2 | 0.1 |
- |
1-benzoyl piperidine |
larger than 0.100 mM |
703559 |
5.3.99.2 | 0.1 |
- |
1-benzoyl-4-(methylsulfonyl)piperazine |
larger than 0.100 mM |
703559 |
5.3.99.2 | 0.1 |
- |
1-phenyl-1-(2-thienyl)methanamine |
larger than 0.100 mM |
703559 |
5.3.99.2 | 7 |
- |
2'-oxo-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]-1',2'-dihydro[2,4'-bipyridine]-5-carboxamide |
at 37°C, pH not specified in the publication |
747270 |
5.3.99.2 | 0.0362 |
- |
2-(2'-benzothiazolyl)-5-styryl-3-(4'-phthalhydrazyl) tetrazolium chloride |
IC50: 0.0362 mM in presence of EDTA, 0.0981 in presence of Mg2+ |
662057 |
5.3.99.2 | 0.000021 |
- |
2-phenyl-5-(1H-pyrazol-3-yl)-1,3-thiazole |
37°C |
693542 |
5.3.99.2 | 0.0007 |
- |
2-phenyl-5-(1H-pyrazol-3-yl)thiazole |
in 0.1 M Tris-HCl, pH 8.0, at 25°C |
715845 |
5.3.99.2 | 0.00004 |
- |
3-(3-cyclopropyl-1H-pyrazol-4-yl)-N-ethyl-5,7-dihydro-6H-pyrrolo[3,4-b]pyridine-6-carboxamide |
pH and temperature not specified in the publication |
748543 |
5.3.99.2 | 0.017 |
- |
3-(3-cyclopropyl-1H-pyrazol-4-yl)pyridine |
pH and temperature not specified in the publication |
748543 |