EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor  |
Reference |
|---|
   3.4.25.1 | 0.000086 |
0.000194 |
(-)-epigallocatechin-3-gallate |
inhibition of the chymotrypsin-like activity of the proteasome in vitro, pH not specified in the publication, temperature not specified in the publication |
702678 |
| 3.4.25.1 | 0.019 |
- |
(2R,3S)-1,2,3,4-tetrahydronaphthalene-2,3-diyl bis(3,4,5-trihydroxybenzoate) |
for the chymotrypsin-like activity, pH 7.5, 37°C |
702678 |
| 3.4.25.1 | 0.029 |
- |
(2R,3S)-1,2,3,4-tetrahydronaphthalene-2,3-diyl bis(3,5-dihydroxybenzoate) |
for the chymotrypsin-like activity, pH 7.5, 37°C |
702678 |
| 3.4.25.1 | 0.00022 |
- |
1-[1-(1-[(2,4-dioxoimidazolidin-1-ylimino)-methyl]-2-phenyl-ethylcarbamoyl)-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-(1H-indol) |
pH 7.5, 30°C |
711621 |
| 3.4.25.1 | 0.85 |
- |
acetyl-Leu-Leu-Arg |
IC50: 0.85 mM for chymotrypsin-like activity, 0.0056 mM for trypsin-like activity |
650902 |
| 3.4.25.1 | 0.11 |
- |
benzyloxycarbonyl-Leu-Gly-Arg |
IC50: 0.11 mM for chymotrypsin-like activity, 0.0066 mM for trypsin-like activity |
650902 |
| 3.4.25.1 | 0.056 |
- |
Benzyloxycarbonyl-Leu-Leu-Arg |
IC50: 0.056 mM for chymotrypsin-like activity, 0.0014 mM for trypsin-like activity |
650902 |
| 3.4.25.1 | 0.017 |
- |
benzyloxycarbonyl-Leu-Ser-Arg |
IC50: 0.017 mM for chymotrypsin-like activity, 0.0017 mM for trypsin-like activity |
650902 |
| 3.4.25.1 | 0.065 |
- |
benzyloxycarbonyl-Leu-Thr-Arg |
IC50: 0.065 mM for chymotrypsin-like activity, 0.0021 mM for trypsin-like activity |
650902 |
| 3.4.25.1 | 0.0089 |
- |
benzyloxycarbonyl-Phe-Ser-Arg |
IC50: 0.0089 mM for chymotrypsin-like activity, 0.002 mM for trypsin-like activity |
650902 |
