EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor  |
Reference |
|---|
   3.4.24.B10 | 0.00593 |
- |
(2R)-N4-hydroxy-N1-[(1S)-1-(1H-indol-3-ylmethyl)-2-(methylamino)-2-oxoethyl]-2-(2-methylpropyl)butanediamide |
IC50: 5930 nM |
667947 |
| 3.4.24.B10 | 0.000025 |
- |
batimastat |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
| 3.4.24.B10 | 0.000028 |
- |
batimastat |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
| 3.4.24.B10 | 0.0011 |
- |
GM6001 |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
| 3.4.24.B10 | 0.0021 |
- |
GM6001 |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
| 3.4.24.B10 | 0.00043 |
- |
marimastat |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
| 3.4.24.B10 | 0.00067 |
- |
marimastat |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
| 3.4.24.B10 | 0.0006 |
- |
MMP inhibitor III |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
| 3.4.24.B10 | 0.0011 |
- |
MMP inhibitor III |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
| 3.4.24.B10 | 0.00012 |
- |
MMP inhibitor V |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
