EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.23.5 | 0.0000000783 |
- |
Tb-9 |
at pH 3.5 and 25°C |
754470 |
3.4.23.5 | 0.000000126 |
- |
TB-11 |
at pH 3.5 and 25°C |
754470 |
3.4.23.5 | 0.000000182 |
- |
tasiamide B |
at pH 3.5 and 25°C |
754470 |
3.4.23.5 | 0.000000693 |
- |
pepstatin A |
at pH 3.5 and 25°C |
754470 |
3.4.23.5 | 0.00000329 |
- |
methyl (5S,8S,11S,12S,16S,19S,22R)-8-(3-amino-3-oxopropyl)-11,22-dibenzyl-12-hydroxy-7,19,21-trimethyl-16-(2-methylpropyl)-3,6,9,14,17,20-hexaoxo-1-phenyl-5-(propan-2-yl)-2-oxa-4,7,10,15,18,21-hexaazatricosan-23-oate |
at pH 3.5 and 25°C |
754470 |
3.4.23.5 | 0.000027 |
- |
(5S,8S,11S,12S,16S,19S,22R)-8-(3-amino-3-oxopropyl)-11,22-dibenzyl-12-hydroxy-7,19,21-trimethyl-16-(2-methylpropyl)-3,6,9,14,17,20-hexaoxo-1-phenyl-5-(propan-2-yl)-2-oxa-4,7,10,15,18,21-hexaazatricosan-23-oic acid |
at pH 3.5 and 25°C |
754470 |
3.4.23.5 | 0.000102 |
- |
methyl (5S,8S,11S,12S,16S,19S)-8-(3-amino-3-oxopropyl)-11-benzyl-12-hydroxy-7,19-dimethyl-16-(2-methylpropyl)-3,6,9,14,17-pentaoxo-1-phenyl-5-(propan-2-yl)-2-oxa-4,7,10,15,18-pentaazaicosan-20-oate |
at pH 3.5 and 25°C |
754470 |
3.4.23.5 | 0.000108 |
- |
(5S,8S,11S,12S,16S,19S)-8-(3-amino-3-oxopropyl)-11-benzyl-12-hydroxy-7,19-dimethyl-16-(2-methylpropyl)-3,6,9,14,17-pentaoxo-1-phenyl-5-(propan-2-yl)-2-oxa-4,7,10,15,18-pentaazaicosan-20-oic acid |
at pH 3.5 and 25°C |
754470 |
3.4.23.5 | 0.000131 |
- |
(6S,9S,12S,13S,17S,20S,23R)-9-(3-amino-3-oxopropyl)-12,23-dibenzyl-13-hydroxy-2,2,8,20,22-pentamethyl-17-(2-methylpropyl)-4,7,10,15,18,21-hexaoxo-6-(propan-2-yl)-3-oxa-5,8,11,16,19,22-hexaazatetracosan-24-oic acid |
at pH 3.5 and 25°C |
754470 |
3.4.23.5 | 0.00019 |
- |
methyl (6S,9S,12S,13S,17S,20S,23R)-9-(3-amino-3-oxopropyl)-12,23-dibenzyl-13-hydroxy-2,2,8,20,22-pentamethyl-17-(2-methylpropyl)-4,7,10,15,18,21-hexaoxo-6-(propan-2-yl)-3-oxa-5,8,11,16,19,22-hexaazatetracosan-24-oate |
at pH 3.5 and 25°C |
754470 |