EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   3.4.22.59 | 0.000011 |
- |
N-[(2R)-1-(3-cyanophenyl)-3-hydroxypropan-2-yl]-5-(3,4-dimethoxyphenyl)furan-3-carboxamide |
in 50 mM HEPES (pH 7.0), 25 mM MgSO4, 0.5 mM EGTA, 5 mM glutathione, 0.01% (v/v) Triton X-100 containing 0.1% (w/v) bovine gamma-globulin, at 22°C |
732713 |
| 3.4.22.59 | 0.0000162 |
- |
Ac-VEID-CHO |
pH 7.2, 37°C, recombinant enzyme |
718301 |
| 3.4.22.59 | 0.0000305 |
- |
Ac-DEVD-CHO |
pH 7.2, 37°C, recombinant enzyme |
718301 |
| 3.4.22.59 | 0.0000532 |
- |
Ac-IETD-CHO |
pH 7.2, 37°C, recombinant enzyme |
718301 |
| 3.4.22.59 | 0.0001286 |
- |
Z-VEID-fluoromethylketone |
pH 7.2, 37°C, recombinant enzyme |
718301 |
| 3.4.22.59 | 0.000151 |
- |
[1-benzyl-2-oxo-5-(thiomorpholin-4-ylsulfonyl)-1,2-dihydro-3H-indol-3-ylidene]propanedinitrile |
- |
699459 |
| 3.4.22.59 | 0.000156 |
- |
[5-(azetidin-1-ylsulfonyl)-1-benzyl-2-oxo-1,2-dihydro-3H-indol-3-ylidene]propanedinitrile |
- |
699459 |
| 3.4.22.59 | 0.000188 |
- |
[1-(4-methoxybenzyl)-2-oxo-5-(thiomorpholin-4-ylsulfonyl)-1,2-dihydro-3H-indol-3-ylidene]propanedinitrile |
- |
699459 |
| 3.4.22.59 | 0.000197 |
- |
[5-(azetidin-1-ylsulfonyl)-1-(4-methoxybenzyl)-2-oxo-1,2-dihydro-3H-indol-3-ylidene]propanedinitrile |
- |
699459 |
| 3.4.22.59 | 0.00023 |
- |
[1-(3,4-dichlorobenzyl)-2-oxo-5-(thiomorpholin-4-ylsulfonyl)-1,2-dihydro-3H-indol-3-ylidene]propanedinitrile |
- |
699459 |
