EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   3.1.1.8 | -999 |
- |
more |
- |
682916, 691944 |
| 3.1.1.8 | 0.00000103 |
- |
(+/-)-N-((1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl)methyl)-N-(2-(dimethylamino)ethyl)-2-naphthamide |
pH 8.0, 25°C |
751285 |
| 3.1.1.8 | 0.0000018 |
- |
(3aS)-3a,8-dimethyl-1-(2-phenylethyl)-1,2,3,3a,8,8a-hexahydropyrrolo[2,3-b]indol-5-yl (cyclohexylmethyl)carbamate |
pH not specified in the publication, at 37°C |
714407 |
| 3.1.1.8 | 0.000003 |
- |
4-methyl-N-(4-(8,9,10,11-tetrahydro-6H-azocino-[2,1-b]quinazolin-13(7H)-ylideneamino)butyl)-N-(3-(8,9,-10,11-tetrahydro-6H-azocino[2,1-b]quinazolin-13(7H)-ylideneamino)propyl)pentanamide |
in 100 mM potassium dihydrogen phosphate buffer, pH 8.0, at 25°C |
714458 |
| 3.1.1.8 | 0.0000034 |
- |
eserine |
pH 7.4, 22°C |
692056 |
| 3.1.1.8 | 0.000004 |
- |
N-(4-(2,3-dihydropyrrolo[2,1-b]quinazolin-9(1H)-ylideneamino)butyl)-N-(3-(2,3-dihydropyrrolo[2,1-b]quinazolin-9(1H)-ylideneamino)propyl)acetamide |
in 100 mM potassium dihydrogen phosphate buffer, pH 8.0, at 25°C |
714458 |
| 3.1.1.8 | 0.0000043 |
- |
(2xi)-1,4:3,6-dianhydro-2-O-(benzylcarbamoyl)-5-O-(phenoxycarbonyl)-D-arabino-hexitol |
pH 7.4, 37°C |
693570 |
| 3.1.1.8 | 0.00000479 |
- |
Carbaryl |
pH 7.4, 25°C, versus propionylthiocholine |
679345 |
| 3.1.1.8 | 0.0000048 |
- |
(9E,9'Z)-N,N'-heptane-1,7-diylbis(2,3-dihydropyrrolo[2,1-b]quinazolin-9(1H)-imine) |
pH and temperature not specified in the publication |
714458 |
| 3.1.1.8 | 0.0000048 |
- |
Carbaryl |
versus propionylthiocholine |
679344 |
