EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.7.7.64 | 0.0404 |
0.0463 |
ethyl 2,4-dimethyl-5-[(2R)-2-[4-(2-phenoxyethyl)piperazin-1-yl]propanoyl]-1H-pyrrole-3-carboxylate |
wild-type enzyme, pH 8.0, 25°C |
761959 |
2.7.7.64 | 0.0472 |
0.0664 |
methyl (2R)-2-[[2-(4-fluorophenyl)sulfanylacetyl]amino]-3-hydroxypropanoate |
wild-type enzyme, pH 8.0, 25°C |
761959 |
2.7.7.64 | 0.0781 |
0.1066 |
(3R)-1-(4-chlorobenzoyl)-N-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)piperidine-3-carboxamide |
wild-type enzyme, pH 8.0, 25°C |
761959 |
2.7.7.64 | 0.135 |
0.175 |
2-[3-(trifluoromethyl)anilino]-1,3-thiazol-4-one |
wild-type enzyme, pH 8.0, 25°C |
761959 |
2.7.7.64 | 0.1698 |
0.1948 |
2-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)oxybenzamide |
wild-type enzyme, pH 8.0 25°C |
761959 |
2.7.7.64 | 0.25 |
- |
2-(furan-2-yl)-N'-(indol-3-ylidenemethyl)quinoline-4-carbohydrazide |
above, wild-type enzyme, pH 8.0, 25°C |
761959 |
2.7.7.64 | 0.25 |
- |
2-[(3As,7aR)-1,3-dioxo-3a,4,7,7a-tetrahydroisoindol-2-yl]-N-[4-(propan-2-ylsulfamoyl)phenyl]acetamide |
above, wild-type enzyme, pH 8.0, 25°C |
761959 |