EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.7.4.9 | 0.0000001 |
- |
2-(3-bromophenoxy)-4-((R)-1-((S)-3-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)piperidin-1-yl)hexyl)benzoic acid |
IC50 below 0.1 nM, pH and temperature not specified in the publication |
722918 |
2.7.4.9 | 0.0000001 |
- |
2-(3-bromophenoxy)-4-(R)-(2-(1-adamantane)-1-((S)-3-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)piperidin-1-yl)ethyl)benzoic acid |
pH and temperature not specified in the publication |
722918 |
2.7.4.9 | 0.0000001 |
- |
2-(3-chlorophenoxy)-4-((R)-1-((S)-3-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)piperidin-1-yl)-2-(tetrahydro-2H-pyran-4-yl)ethyl)benzoic acid |
IC50 below 0.1 nM, pH and temperature not specified in the publication |
722918 |
2.7.4.9 | 0.0000001 |
- |
2-(3-chlorophenoxy)-4-((R)-2-cyclohexyl-1-((S)-3-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)piperidin-1-yl)ethyl)benzoic acid |
IC50 below 0.1 nM, pH and temperature not specified in the publication |
722918 |
2.7.4.9 | 0.0000001 |
- |
2-(3-chlorophenoxy)-4-((R)-3-ethyl-1-((S)-3-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)piperidin-1-yl)pentyl)benzoic acid |
pH and temperature not specified in the publication |
722918 |
2.7.4.9 | 0.0000002 |
- |
2-(3-chlorophenoxy)-4-((S)-1-((S)-3-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)piperidin-1-yl)butyl)benzoic acid |
IC50 below 0.2 nM, pH and temperature not specified in the publication |
722918 |
2.7.4.9 | 0.0000002 |
- |
2-(3-chlorophenoxy)-4-((S)-3-methyl-1-((S)-3-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)piperidin-1-yl)butyl)benzoic acid |
pH and temperature not specified in the publication |
722918 |
2.7.4.9 | 0.0000002 |
- |
TK-666 |
pH and temperature not specified in the publication |
722918 |
2.7.4.9 | 0.0000003 |
- |
(3-chlorophenoxy)-4-((S)-1-((S)-3-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)piperidin-1-yl)propyl)benzoic acid |
pH and temperature not specified in the publication |
722918 |
2.7.4.9 | 0.0000003 |
- |
2-(3-bromophenoxy)-4-((R)-3-ethyl-3-methyl-1-((S)-3-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)piperidin-1-yl)pentyl)benzoic acid |
pH and temperature not specified in the publication |
722918 |