EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.7.11.15 | 0.0000041 |
- |
RNA aptamer C13 |
inhibition of GRK2, kinetics, overview |
690032 |
2.7.11.15 | 0.000006 |
- |
3-(3-methoxybenzyl)-6-(1H-pyrazol-4-yl)quinazolin-4(3H)-one |
pH and temperature not specified in the publication |
760708 |
2.7.11.15 | 0.000009 |
- |
N-(4-fluorophenyl)-3-[[4-oxo-6-(1H-pyrazol-4-yl)quinazolin-3(4H)-yl]methyl]benzamide |
pH and temperature not specified in the publication |
760708 |
2.7.11.15 | 0.00001 |
- |
N-[(2,6-difluorophenyl)methyl]-3-[[4-oxo-6-(1H-pyrazol-4-yl)quinazolin-3(4H)-yl]methyl]benzamide |
IC50 below 0.00001 mM, pH and temperature not specified in the publication |
760708 |
2.7.11.15 | 0.00001 |
- |
N-[(4-fluorophenyl)methyl]-3-[[4-oxo-6-(1H-pyrazol-4-yl)quinazolin-3(4H)-yl]methyl]benzamide |
IC50 below 0.00001 mM, pH and temperature not specified in the publication |
760708 |
2.7.11.15 | 0.000012 |
- |
3-[1-(3-methoxyphenyl)-3-(methylamino)propyl]-6-(1H-pyrazol-4-yl)quinazolin-4(3H)-one |
pH and temperature not specified in the publication |
760708 |
2.7.11.15 | 0.000013 |
- |
3-[(1R)-1-(3-methoxyphenyl)ethyl]-6-(1H-pyrazol-4-yl)quinazolin-4(3H)-one |
pH and temperature not specified in the publication |
760708 |
2.7.11.15 | 0.000018 |
- |
3-(4-fluoro-3-methoxybenzyl)-6-(1H-pyrazol-4-yl)quinazolin-4(3H)-one |
pH and temperature not specified in the publication |
760708 |
2.7.11.15 | 0.000019 |
- |
2-(3-methoxybenzyl)-7-(1H-pyrazol-4-yl)phthalazin-1(2H)-one |
pH and temperature not specified in the publication |
760708 |
2.7.11.15 | 0.00002 |
- |
Takeda103A |
at pH 7.0, temperature not specified in the publication |
738847 |