EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
    2.7.1.145 | 0.00257 |
- |
(E)-5-(2-bromovinyl)-2'-deoxyuridine |
IC50: 0.00257 mM for reaction with thymidine and 0.00194 mM for reaction with 2'-deoxycytidine |
636841 |
| 2.7.1.145 | 0.0026 |
- |
(E)-5-(2-bromovinyl)-2'-deoxyuridine 5'-monophosphate |
IC50: 0.0026 mM, reaction with thymidine, fusion protein with glutathione S-transferase |
636843 |
| 2.7.1.145 | 0.0069 |
- |
(E)-5-(2-bromovinyl)-2'-deoxyuridine 5'-triphosphate |
IC50: 0.0069 mM, reaction with thymidine, fusion protein with glutathione S-transferase. The inhibitor is efficiently metabolized to its 5'-mono-, 5'-di- and 5'-triphosphate derivatives in the insect cell culture and abundently incorporated into the insec |
636843 |
| 2.7.1.145 | 0.012 |
- |
dTTP |
IC50: 0.012 mM, reaction with thymidine, fusion protein with glutathione S-transferase |
636843 |
| 2.7.1.145 | 0.0163 |
- |
1-(2-deoxy-2-fluoro-beta-D-arabinofuranosyl)-5-iodouracil |
IC50: 0.0163 mM for reaction with thymidine and 0.0154 mM for reaction with 2'-deoxycytidine |
636841 |
| 2.7.1.145 | 0.0258 |
- |
5-fluoro-2'-deoxyuridine |
IC50: 0.0258 mM for reaction with thymidine and 0.02235 mM for reaction with 2'-deoxycytidine |
636841 |
| 2.7.1.145 | 0.0277 |
- |
(E)-5-(2-bromovinyl)-1-beta-D-arabinofuranosyluracil |
IC50: 0.0277 mM for reaction with thymidine and 0.0158 mM for reaction with 2'-deoxycytidine |
636841 |
| 2.7.1.145 | 0.0419 |
- |
3'-azido-2',3'-dideoxythymidine |
IC50: 0.0419 mM for reaction with thymidine and 0.0296 mM for reaction with 2'-deoxycytidine |
636841 |
| 2.7.1.145 | 0.0534 |
- |
1-beta-D-arabinofuranosylcytosine |
IC50: 0.0534 mM for reaction with thymidine and 0.089 mM for reaction with 2'-deoxycytidine |
636841 |
| 2.7.1.145 | 0.057 |
- |
1-beta-D-arabinofuranosyluracil |
IC50: 0.057 mM for reaction with thymidine and 0.058 mM for reaction with 2'-deoxycytidine |
636841 |
