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Results 1 - 10 of 32 > >>
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EC Number IC50 Value IC50 Value Maximum Inhibitor Commentary Reference
Display the word mapDisplay the reaction diagram Show all sequences 2.5.1.60-999 - more chemicals that cause an activity decrease of more than 70% at 100 microM are selected for inhibition studies 709461
Display the word mapDisplay the reaction diagram Show all sequences 2.5.1.60-999 - more the inhibitory action of 2-hydroxy-2-phosphono-3-pyridin-3-yl-propionic acid with substrates Rab1a-CSC and Rab1a-CCS are not determined, and is not significant (IC50 > 2 mM) with the substrates Rab1a-CS, Rab1aSC, Rab27a-CVLS, Rab5a-CCQNI, Rab5a-CVLL, Rab13-CSLG (wild type), Rab18-CSVL (wild type), and Rab23-CSVP (wild type), and IC50 > 1.592 mM with Rab6a-CSC 709077
Display the word mapDisplay the reaction diagram Show all sequences 2.5.1.600.0021 - (2R,3R,4S,5R)-2-(4-bromophenyl)-4-(hexylsulfanyl)-1-[(4-methylphenyl)sulfonyl]-5-propylpyrrolidine-3-carboxylic acid - 687811
Display the word mapDisplay the reaction diagram Show all sequences 2.5.1.600.0022 - (2R,3R,4S,5R)-2-(4-bromophenyl)-5-hexyl-4-(hexylsulfanyl)-1-[(4-methylphenyl)sulfonyl]pyrrolidine-3-carboxylic acid - 687811
Display the word mapDisplay the reaction diagram Show all sequences 2.5.1.600.0031 - (2R,3R,4S,5R)-4-[(3-tert-butoxy-3-oxopropyl)sulfanyl]-2-(4-chlorophenyl)-1-[(4-chlorophenyl)sulfonyl]-5-(cyclopentylmethyl)pyrrolidine-3-carboxylic acid - 687811
Display the word mapDisplay the reaction diagram Show all sequences 2.5.1.600.0036 - (2R,3R,4S,5R)-2-(4-bromophenyl)-1-[(4-methylphenyl)sulfonyl]-4-(pentylsulfanyl)-5-propylpyrrolidine-3-carboxylic acid - 687811
Display the word mapDisplay the reaction diagram Show all sequences 2.5.1.600.0041 - N-[(benzyloxy)carbonyl]-D-tyrosyl-L-phenylalanyl-L-tyrosine most potent of the class I inhibitors (compounds possessing a free carboxylic or hydroxamic acid at the C-terminus and lipophilic N-termini), 9 microM (3,7,11-trimethyl-12-(7-nitrobenzo[1,2,5]oxadiazo-4-ylamino)-dodeca-2,6,19-trien-1) diphosphate, 3 microM Rab7, 3 microM Rab escort protein, 400 nM enzyme 709461
Display the word mapDisplay the reaction diagram Show all sequences 2.5.1.600.0045 - (2R,3R,4S,5R)-2-(4-bromophenyl)-4-[(4-methoxyphenyl)sulfanyl]-1-[(4-methylphenyl)sulfonyl]-5-propylpyrrolidine-3-carboxylic acid - 687811
Display the word mapDisplay the reaction diagram Show all sequences 2.5.1.600.0047 - (2R,3R,4S,5R)-4-[(3-tert-butoxy-3-oxopropyl)sulfanyl]-2-(3-chlorophenyl)-5-(cyclopentylmethyl)-1-[(4-methylphenyl)sulfonyl]pyrrolidine-3-carboxylic acid - 687811
Display the word mapDisplay the reaction diagram Show all sequences 2.5.1.600.0048 - (2R,3R,4S,5R)-2-(4-bromophenyl)-5-ethyl-4-(hexylsulfanyl)-1-[(4-methylphenyl)sulfonyl]pyrrolidine-3-carboxylic acid - 687811
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