EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.14.14.74 | 0.00015 |
- |
terfenadone |
substrate astemizole, liver microsome, pH 7.4, 37°C |
744774 |
1.14.14.74 | 0.00031 |
- |
terfenadone |
substrate albendazole, liver microsome, pH 7.4, 37°C |
744774 |
1.14.14.74 | 0.00195 |
- |
danazol |
substrate ebastine, liver microsome, pH 7.4, 37°C |
744774 |
1.14.14.74 | 0.0021 |
- |
terfenadone |
substrate terfenadine, liver microsome, pH 7.4, 37°C |
744774 |
1.14.14.74 | 0.00214 |
- |
danazol |
substrate terfenadine, liver microsome, pH 7.4, 37°C |
744774 |
1.14.14.74 | 0.004 |
- |
hydroxyebastine |
substrate terfenadine, liver microsome, pH 7.4, 37°C |
744774 |
1.14.14.74 | 0.00427 |
- |
terfenadone |
substrate ebastine, liver microsome, pH 7.4, 37°C |
744774 |
1.14.14.74 | 0.00928 |
- |
hydroxyebastine |
substrate astemizole, liver microsome, pH 7.4, 37°C |
744774 |
1.14.14.74 | 0.0111 |
- |
hydroxyebastine |
substrate albendazole, liver microsome, pH 7.4, 37°C |
744774 |
1.14.14.74 | 0.0138 |
- |
danazol |
substrate albendazole, liver microsome, pH 7.4, 37°C |
744774 |