EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.14.11.66 | 0.079 |
- |
(R)-2-hydroxyglutarate |
pH and temperature not specified in the publication |
756531 |
1.14.11.66 | 0.097 |
- |
(S)-2-hydroxyglutarate |
pH and temperature not specified in the publication |
756531 |
1.14.11.66 | 0.037 |
- |
2-(2-((chroman-6-ylmethyl)amino)pyrimidin-4-yl)isonicotinic acid |
pH 7.5, 37°C, recombinant enzyme |
744722 |
1.14.11.66 | 0.003 |
- |
3-(9-(dimethylamino)-N-hydroxynonanamido)propanoic acid |
pH 7.5, 37°C, recombinant enzyme |
744722 |
1.14.11.66 | 0.2 |
- |
3-[hydroxy-[5-[[(1R)-2-(hydroxyamino)-2-oxo-1-[(4-phenylphenyl)methyl]ethyl]amino]-5-oxo-pentanoyl]amino]propanoic acid |
pH 7.5, 37°C, recombinant enzyme |
744722 |
1.14.11.66 | 0.0703 |
- |
3-[hydroxy-[5-[[(1S)-2-(hydroxyamino)-2-oxo-1-[(4-phenylphenyl)methyl]ethyl]amino]-5-oxo-pentanoyl]amino]propanoic acid |
pH 7.5, 37°C, recombinant enzyme |
744722 |
1.14.11.66 | 0.0606 |
- |
3-[hydroxy-[7-[[(1S)-2-methoxy-2-oxo-1-[(4-phenylphenyl)methyl]ethyl]amino]-7-oxo-heptanoyl]amino]propanoic acid |
pH 7.5, 37°C, recombinant enzyme |
744722 |
1.14.11.66 | 0.0068 |
- |
3-[hydroxy-[8-[[(1R)-2-(hydroxyamino)-2-oxo-1-[(4-phenylphenyl)methyl]ethyl]amino]-8-oxo-octanoyl]amino]propanoic acid |
pH 7.5, 37°C, recombinant enzyme |
744722 |
1.14.11.66 | 0.0136 |
- |
3-[hydroxy-[8-[[(1S)-2-(hydroxyamino)-2-oxo-1-[(4-phenylphenyl)methyl]ethyl]amino]-8-oxo-octanoyl]amino]propanoic acid |
pH 7.5, 37°C, recombinant enzyme |
744722 |
1.14.11.66 | 0.0371 |
- |
3-[hydroxy-[8-[[(1S)-2-methoxy-2-oxo-1-[(4-phenylphenyl)methyl]ethyl]amino]-8-oxo-octanoyl]amino]propanoic acid |
pH 7.5, 37°C, recombinant enzyme |
744722 |