EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.1.5.3 | 0.0006 |
- |
6-(7-nitro-2,1,3-benzoxadiazol-4-ylthio)hexanol |
at pH 7.5 and 25°C |
740482 |
1.1.5.3 | 0.0007 |
0.001 |
4-[4-(1H-naphtho[2,3-d]imidazol-2-yl)anilino]-4-oxobutanoic acid |
pH not specified in the publication, 37°C |
741302 |
1.1.5.3 | 0.0019 |
- |
metronidazole |
at pH 7.5 and 25°C |
740482 |
1.1.5.3 | 0.003 |
- |
4-[4-[5-(cyclohexa-2,4-diene-1-carbonyl)-1H-benzimidazol-2-yl]anilino]-4-oxobutanoic acid |
pH not specified in the publication, 37°C |
741302 |
1.1.5.3 | 0.005 |
- |
4-[4-(5-methyl-1H-benzimidazol-2-yl)anilino]-4-oxobutanoic acid |
pH not specified in the publication, 37°C |
741302 |
1.1.5.3 | 0.0063 |
0.008 |
4-[4-(1H-benzimidazol-2-yl)anilino]-4-oxobutanoic acid |
pH not specified in the publication, 37°C |
741302 |
1.1.5.3 | 0.015 |
- |
4-[4-(1,3-benzothiazol-2-yl)anilino]-4-oxobutanoic acid |
pH not specified in the publication, 37°C |
741302 |
1.1.5.3 | 0.02 |
- |
4-[4-(1,3-benzoxazol-2-yl)anilino]-4-oxobutanoic acid |
pH not specified in the publication, 37°C |
741302 |
1.1.5.3 | 0.05 |
- |
4-[3-(1H-benzimidazol-2-yl)anilino]-4-oxobutanoic acid |
pH not specified in the publication, 37°C |
741302 |
1.1.5.3 | 0.08 |
- |
N-[4-(5,6-dihydro-1H-benzimidazol-2-yl)phenyl]furan-2-carboxamide |
pH not specified in the publication, 37°C |
741302 |