EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
    5.3.99.2 | 0.000075 |
- |
N-[4-methyl-3-[([3-[(4-methylpiperazin-1-yl)methyl]phenyl]carbonyl)amino]phenyl]-3-phenylisothiazole-5-carboxamide |
37°C |
693542 |
| 5.3.99.2 | 0.00013 |
- |
N-[5-(1H-indol-4-yl)pyridin-3-yl]-3-(piperidin-1-yl)propanamide |
at 37°C, pH not specified in the publication |
747270 |
| 5.3.99.2 | 0.000138 |
- |
4-[[4-(4-fluoro-3-methylphenyl)-1,3-thiazol-2-yl]amino]-2-hydroxybenzoic acid |
37°C |
693542 |
| 5.3.99.2 | 0.00018 |
- |
4-(dimethylamino)-N-[5-(1H-indol-4-yl)pyridin-3-yl]butanamide |
at 37°C, pH not specified in the publication |
747270 |
| 5.3.99.2 | 0.0002 |
- |
Cibacron blue 3GA |
- |
703559 |
| 5.3.99.2 | 0.0002 |
- |
erythrosine sodium |
at pH 6.5 and 30°C |
747503 |
| 5.3.99.2 | 0.00023 |
- |
6-(pyrrolidin-1-yl)-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]pyridine-3-carboxamide |
at 37°C, pH not specified in the publication |
747270 |
| 5.3.99.2 | 0.0003 |
- |
3-acetamido-N-[5-(1H-indol-4-yl)pyridin-3-yl]propanamide |
at 37°C, pH not specified in the publication |
747270 |
| 5.3.99.2 | 0.0003 |
- |
suramin |
at pH 6.5 and 30°C |
747503 |
| 5.3.99.2 | 0.00032 |
- |
6-(morpholin-4-yl)-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]pyridine-3-carboxamide |
at 37°C, pH not specified in the publication |
747270 |
