5.3.99.2 0.000021 - 2-phenyl-5-(1H-pyrazol-3-yl)-1,3-thiazole 37°C 693542 5.3.99.2 0.000026 - N-[5-(1H-indol-4-yl)pyridin-3-yl]-3-(pyridin-3-yl)propanamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.000031 - 6-phenoxy-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]pyridine-3-carboxamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.000032 - N-[5-(1H-indol-4-yl)pyridin-3-yl]propanamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.000035 - N-[5-(1H-indol-4-yl)pyridin-3-yl]-5-oxopyrrolidine-2-carboxamide (incorrect configuration definition!) at 37°C, pH not specified in the publication 747270 5.3.99.2 0.00004 - 3-(3-cyclopropyl-1H-pyrazol-4-yl)-N-ethyl-5,7-dihydro-6H-pyrrolo[3,4-b]pyridine-6-carboxamide pH and temperature not specified in the publication 748543 5.3.99.2 0.000043 - N-[5-(1H-indol-4-yl)pyridin-3-yl]-2-(1H-tetrazol-1-yl)acetamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.000048 - 6-(piperidin-1-yl)-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]pyridine-3-carboxamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.00006 - 6-(3-methoxyphenyl)-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]pyridine-3-carboxamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.000071 - 6'-oxo-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]-1',6'-dihydro[2,2'-bipyridine]-5-carboxamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.000075 - N-[4-methyl-3-[([3-[(4-methylpiperazin-1-yl)methyl]phenyl]carbonyl)amino]phenyl]-3-phenylisothiazole-5-carboxamide 37°C 693542 5.3.99.2 0.00013 - N-[5-(1H-indol-4-yl)pyridin-3-yl]-3-(piperidin-1-yl)propanamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.000138 - 4-[[4-(4-fluoro-3-methylphenyl)-1,3-thiazol-2-yl]amino]-2-hydroxybenzoic acid 37°C 693542 5.3.99.2 0.00018 - 4-(dimethylamino)-N-[5-(1H-indol-4-yl)pyridin-3-yl]butanamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.0002 - Cibacron blue 3GA - 703559 5.3.99.2 0.0002 - erythrosine sodium at pH 6.5 and 30°C 747503 5.3.99.2 0.00023 - 6-(pyrrolidin-1-yl)-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]pyridine-3-carboxamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.0003 - 3-acetamido-N-[5-(1H-indol-4-yl)pyridin-3-yl]propanamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.0003 - suramin at pH 6.5 and 30°C 747503 5.3.99.2 0.00032 - 6-(morpholin-4-yl)-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]pyridine-3-carboxamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.0004 - Tannic acid at pH 6.5 and 30°C 747503 5.3.99.2 0.0005 - N-cyclopentyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine pH and temperature not specified in the publication 748543 5.3.99.2 0.00059 - 6-(3-oxopiperazin-1-yl)-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]pyridine-3-carboxamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.0006 - sanguinarine sulfate at pH 6.5 and 30°C 747503 5.3.99.2 0.0007 - 2-phenyl-5-(1H-pyrazol-3-yl)thiazole in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.0007 - N-benzhydryl-5-(3-hydroxyphenyl)thiophene-2-carboxamide in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.00092 - 3-phenyl-5-(1H-pyrazol-3-yl)-1,2-oxazole 37°C 693542 5.3.99.2 0.001 - N-(1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-yl)-3'-hydroxybiphenyl-4-carboxamide in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.0012 - N-(1-amino-1-oxo-3-phenylpropan-2-yl)-6-(thiophen-2-yl)nicotinamide in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.0012 - N-[5-(1H-indol-4-yl)pyridin-3-yl]-2-(1-methyl-1H-imidazol-5-yl)acetamide at 37°C, pH not specified in the publication 747270 5.3.99.2 0.0013 - N-(1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl)-5-(3-hydroxyphenyl)thiophene-2-carboxamide in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.0014 - 4-[[4-(4-fluoro-3-methylphenyl)-1,3-thiazol-2-yl]amino]-2-hydroxybenzoic acid in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.0017 - chlorophyllide copper complex sodium salt at pH 6.5 and 30°C 747503 5.3.99.2 0.0018 - HQL-79 - 703559 5.3.99.2 0.0018 - iopanic acid at pH 6.5 and 30°C 747503 5.3.99.2 0.0019 - 5-(3-aminophenyl)-N-benzhydrylthiophene-2-carboxamide in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.002 - montelukast sodium at pH 6.5 and 30°C 747503 5.3.99.2 0.0021 - N-(1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-yl)-5-(3-hydroxyphenyl)thiophene-2-carboxamide in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.003 - 4-dibenzo [a,d]cyclohepten-5-ylidene-1-[4-(2H-tetrazol-5-yl)-butyl]-piperidine inhibition of enzyme in lipocalin-type prostaglandin-D synthase-expressing TE-671 cells after stimulation with Ca2+-ionophore A23187 693254 5.3.99.2 0.0033 - merbromin at pH 6.5 and 30°C 747503 5.3.99.2 0.0037 - N-(1-amino-1-oxo-3-phenylpropan-2-yl)-5-(3-hydroxyphenyl)-thiophene-2-carboxamide in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.0038 - HQL-79 in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.0046 - N-(1-amino-1-oxo-3-phenylpropan-2-yl)-3'-hydroxybiphenyl-4-carboxamide in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.0055 - candesartan cilextil at pH 6.5 and 30°C 747503 5.3.99.2 0.0059 - HQL-79 pH and temperature not specified in the publication 713649 5.3.99.2 0.0071 - N-(1-amino-4-methyl-1-oxopentan-2-yl)-5-(3-hydroxyphenyl)-thiophene-2-carboxamide in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.008 - N-(2-amino-2-oxoethyl)-5-(3-hydroxyphenyl)thiophene-2-carboxamide in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.0084 - epirubicin hydrochloride at pH 6.5 and 30°C 747503 5.3.99.2 0.0085 - N-cyclopentyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine pH and temperature not specified in the publication 748543 5.3.99.2 0.0086 - deoxycorticosterone acetate at pH 6.5 and 30°C 747503 5.3.99.2 0.0089 - Hexachlorophene at pH 6.5 and 30°C 747503 5.3.99.2 0.0092 - NSC4502 - 703559 5.3.99.2 0.0108 - N-(diphenylmethyl)-2-(3-hydroxyphenyl)-1,3-thiazole-4-carboxamide in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.0114 - phenyl-(3-thienyl)-methanone - 703559 5.3.99.2 0.012 - bithionate sodium at pH 6.5 and 30°C 747503 5.3.99.2 0.0128 - phenyl(thiophen-2-yl)methanone in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.0132 - bromocriptine mesylate at pH 6.5 and 30°C 747503 5.3.99.2 0.0134 - fluorescein at pH 6.5 and 30°C 747503 5.3.99.2 0.0137 - tranilast at pH 6.5 and 30°C 747503 5.3.99.2 0.016 - cyclopentyl-phenylketone - 703559 5.3.99.2 0.017 - 3-(3-cyclopropyl-1H-pyrazol-4-yl)pyridine pH and temperature not specified in the publication 748543 5.3.99.2 0.0172 - pyrvinium pamoate at pH 6.5 and 30°C 747503 5.3.99.2 0.0203 - Ketoprofen at pH 6.5 and 30°C 747503 5.3.99.2 0.0208 - pararosaniline pamoate at pH 6.5 and 30°C 747503 5.3.99.2 0.023 - 5-amino-4-[[(3'-hydroxybiphenyl-4-yl)carbonyl]amino]-5-oxopentanoic acid in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.0237 - anthralin at pH 6.5 and 30°C 747503 5.3.99.2 0.0248 - N-(1-amino-1-oxo-3-phenylpropan-2-yl)-3,3'-dihydroxybiphenyl-4-carboxamide in 0.1 M Tris-HCl, pH 8.0, at 25°C 715845 5.3.99.2 0.027 - Sulfobromophthalein - 703559 5.3.99.2 0.029 - nisoldipine at pH 6.5 and 30°C 747503 5.3.99.2 0.0362 - 2-(2'-benzothiazolyl)-5-styryl-3-(4'-phthalhydrazyl) tetrazolium chloride IC50: 0.0362 mM in presence of EDTA, 0.0981 in presence of Mg2+ 662057 5.3.99.2 0.0393 - sennoside A at pH 6.5 and 30°C 747503 5.3.99.2 0.044 - Ethacrynic acid at pH 6.5 and 30°C 747503 5.3.99.2 0.0622 - benzophenone - 703559 5.3.99.2 0.065 - nocodazole - 703559 5.3.99.2 0.0875 - 3-benzoylpyrrole - 703559 5.3.99.2 0.1 - 1-benzoyl piperazine larger than 0.100 mM 703559 5.3.99.2 0.1 - 1-benzoyl piperidine larger than 0.100 mM 703559 5.3.99.2 0.1 - 1-benzoyl-4-(methylsulfonyl)piperazine larger than 0.100 mM 703559 5.3.99.2 0.1 - 1-phenyl-1-(2-thienyl)methanamine larger than 0.100 mM 703559 5.3.99.2 0.1 - AB179670 larger than 0.100 mM 703559 5.3.99.2 0.1 - CMB5256165 larger than 0.100 mM 703559 5.3.99.2 0.1 - cyclohexyl-phenylketone larger than 0.100 mM 703559 5.3.99.2 0.1 - N-phenyl-2-thiophene-carboxamide larger than 0.100 mM 703559 5.3.99.2 0.1 - phenyl-(2-thienyl)-methanol larger than 0.100 mM 703559 5.3.99.2 0.105 - NSC151248 - 703559 5.3.99.2 0.117 - CMB5190724 - 703559 5.3.99.2 0.1223 - Ethacrynic acid - 703559 5.3.99.2 0.3 - oxfendazole larger than 0.300 mM 703559 5.3.99.2 7 - 2'-oxo-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]-1',2'-dihydro[2,4'-bipyridine]-5-carboxamide at 37°C, pH not specified in the publication 747270