EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.24.B10 | 0.00043 |
- |
marimastat |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
3.4.24.B10 | 0.0006 |
- |
MMP inhibitor III |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
3.4.24.B10 | 0.00067 |
- |
marimastat |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
3.4.24.B10 | 0.001 |
- |
TAPI-1 |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
3.4.24.B10 | 0.0011 |
- |
GM6001 |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
3.4.24.B10 | 0.0011 |
- |
MMP inhibitor III |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
3.4.24.B10 | 0.0014 |
- |
TAPI-1 |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
3.4.24.B10 | 0.0014 |
- |
TAPI-2 |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
3.4.24.B10 | 0.0015 |
- |
MMP-3 inhibitor VIII |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |
3.4.24.B10 | 0.0018 |
- |
TAPI-2 |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C |
733079 |