EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.22.51 | 0.1 |
- |
2-(N-4-methyl-benzylidenehydrazino)-4-trifluoromethyl-pyrimidine |
above 0.1 mM |
696710 |
3.4.22.51 | 0.1 |
- |
2-(N-4-nitro-benzylidenehydrazino)-4-trifluoromethylpyrimidine |
about 0.1 mM |
696710 |
3.4.22.51 | 0.1 |
- |
2-[(benzofuroxan-5-yl)methylene]-1-(4-hydroxybenzylidene)hydrazine |
- |
696729 |
3.4.22.51 | 0.1 |
- |
4-(benzofuroxan-5-ylmethyloxy)benzaldehyde semicarbazone |
above 0.1 mM |
696729 |
3.4.22.51 | 0.1 |
- |
benzofuroxan-5-carboxaldehyde thiosemicarbazone |
above 0.1 mM |
696729 |
3.4.22.51 | 0.1 |
- |
N4-allyl benzofuroxan-5-carboxaldehyde thiosemicarbazone |
above 0.1 mM |
696729 |
3.4.22.51 | 0.15 |
- |
2-(N-2-methoxy-benzylidenehydrazino)-6-methyl-4-trifluoromethyl-pyrimidine |
above 0.15 mM |
696710 |
3.4.22.51 | 0.15 |
- |
2-(N-benzylidenehydrazino)-4-trifluoromethylpyrimidine |
above 0.15 mM |
696710 |
3.4.22.51 | 1.41 |
- |
N-[4-methyl-3-(piperidin-1-ylsulfonyl)phenyl]-4-oxo-4-(3-phenyl-4,5-dihydro-1H-pyrazol-1-yl)butanamide |
23°C, pH 6.5 |
753924 |