EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
    2.7.1.33 | 0.00046 |
- |
N-(benzo[d][1,3]dioxol-5-ylmethyl)pantothenamide |
pH 7.6, 25°C |
758568 |
| 2.7.1.33 | 0.0007 |
- |
WIN 62577 |
isoform PanK3, at pH 7.5 and 37°C |
722018 |
| 2.7.1.33 | 0.00082 |
- |
[[2-[[4-(6-methylpyridin-2-yl)piperazin-1-yl]methyl]-4'-(trifluoromethoxy)biphenyl-4-yl]oxy]acetic acid |
in 50 mM PIPES-NaOH (pH 7.0), 25 mM KCl, 20 mM MgCl, at 25°C |
722830 |
| 2.7.1.33 | 0.00087 |
- |
[2-[(3-chlorophenyl)sulfanyl]quinolin-4-yl](piperidin-1-yl)methanone |
in 50 mM PIPES-NaOH (pH 7.0), 25 mM KCl, 20 mM MgCl, at 25°C |
722830 |
| 2.7.1.33 | 0.001 |
- |
pioglitazone hydrochloride |
isoform PanK3, at pH 7.5 and 37°C |
722018 |
| 2.7.1.33 | 0.0013 |
- |
Reactive blue 2 |
isoform PanK3, at pH 7.5 and 37°C |
722018 |
| 2.7.1.33 | 0.0016 |
- |
ephedrine hydrochloride |
isoform PanK3, at pH 7.5 and 37°C |
722018 |
| 2.7.1.33 | 0.0016 |
- |
Psi-rhodomyrtoxin |
isoform PanK3, at pH 7.5 and 37°C |
722018 |
| 2.7.1.33 | 0.0017 |
- |
rosiglitazone |
isoform PanK3, at pH 7.5 and 37°C |
722018 |
| 2.7.1.33 | 0.0025 |
- |
pregnenolone sulfate |
isoform PanK3, at pH 7.5 and 37°C |
722018 |
