EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.1.2.20 | 0.001 |
- |
N-ethylmaleimide |
- |
646129 |
3.1.2.20 | 0.008 |
- |
CoA |
pH 8.0, 28°C, versus acetyl-CoA |
646180 |
3.1.2.20 | 0.052 |
- |
ATP |
pH 8.0, 28°C, versus acetyl-CoA |
646180 |
3.1.2.20 | 0.053 |
- |
CoA-S-S-CoA |
pH 8.0, 28°C, versus acetyl-CoA |
646180 |
3.1.2.20 | 0.085 |
- |
CoA-S-S-CoA |
pH 8.0, 28°C, with palmitoyl-CoA as substrate |
646180 |
3.1.2.20 | 0.5 |
- |
NADH |
pH 8.0, 28°C, with palmitoyl-CoA as substrate |
646180 |
3.1.2.20 | 0.164 |
- |
Nafamostat |
- |
683004 |
3.1.2.20 | -999 |
- |
more |
noncompetitive inhibition of YciA-catalyzed isobutyryl-CoA hydrolysis is observed which defined a Kii of 0.0047 mM (Vmax altered) and a Kis of 0.33 microM (Vmax/Km altered) |
690932 |
3.1.2.20 | 0.0019 |
- |
hexyl-CoA |
- |
690932 |
3.1.2.20 | 0.0054 |
- |
hexyl-CoA |
- |
690932 |