EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.7.10.2 | -999 |
- |
more |
- |
661458 |
2.7.10.2 | -999 |
- |
more |
substrate inhibition kinetics and analysis |
674905 |
2.7.10.2 | 0.00000011 |
- |
N-(3-[2-[4-(2-acetamidoethoxy)anilino]quinazolin-6-yl]-4-methylphenyl)-3-(trifluoromethyl)benzamide |
non-receptor tyrosine kinase Src, pH and temperature not specified in the publication |
737321 |
2.7.10.2 | 0.00000012 |
- |
N-[3-[2-(cyclopropylamino)quinazolin-6-yl]-4-methylphenyl]-3-(trifluoromethyl)benzamide |
non-receptor tyrosine kinase Abl, pH and temperature not specified in the publication |
737321 |
2.7.10.2 | 0.00000013 |
- |
iclusig |
non-receptor tyrosine kinase Abl, pH and temperature not specified in the publication |
737321 |
2.7.10.2 | 0.00000018 |
- |
N-(3-[2-[4-(2-acetamidoethoxy)anilino]quinazolin-6-yl]-4-methylphenyl)-3-(trifluoromethyl)benzamide |
non-receptor tyrosine kinase Abl, pH and temperature not specified in the publication |
737321 |
2.7.10.2 | 0.00000022 |
- |
N-[4-[4-amino-1-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl]phenyl]-N'-[3-(trifluoromethyl)phenyl]urea |
non-receptor tyrosine kinase Abl, pH and temperature not specified in the publication |
737321 |
2.7.10.2 | 0.00000028 |
- |
N-(4-methyl-3-[[3-(pyrimidin-4-yl)pyridin-2-yl]amino]phenyl)-3-(trifluoromethyl)benzamide |
non-receptor tyrosine kinase Abl, pH and temperature not specified in the publication |
737321 |
2.7.10.2 | 0.00000039 |
- |
N-[4-methyl-3-([3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl]amino)phenyl]-3-(trifluoromethyl)benzamide |
non-receptor tyrosine kinase Abl, pH and temperature not specified in the publication |
737321 |
2.7.10.2 | 0.00000042 |
- |
rebastinib |
non-receptor tyrosine kinase Abl, pH and temperature not specified in the publication |
737321 |