EC Number |
KM Value [mM] |
KM Value Maximum [mM] |
Substrate |
Reference |
---|
2.1.1.374 | 0.0014 |
- |
3-methyl-1-oxo-2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-1,5-dihydrobenzo[4,5]imidazo[1,2-a]pyridine-4-carbonitrile |
pH 7.4, 37°C, mutant enzyme S140A |
760066 |
2.1.1.374 | 0.004 |
- |
3-methyl-1-oxo-2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-1,5-dihydrobenzo[4,5]imidazo[1,2-a]pyridine-4-carbonitrile |
pH 7.4, 37°C, wild-type enzyme |
760066 |
2.1.1.374 | 0.0094 |
- |
2-heptyl-1-hydroxyquinolin-4(1H)-one |
pH 7.0 30°C |
759185 |
2.1.1.374 | 0.0098 |
- |
2-heptyl-1-hydroxyquinolin-4(1H)-one |
pH 7.0 30°C |
759185 |