EC Number |
Inhibitors |
Structure |
---|
1.3.1.9 | (-)-catechin gallate |
IC50: 0.3 microM |
|
1.3.1.9 | (-)-epicatechin gallate |
IC50: 0.2 microM |
|
1.3.1.9 | (-)-epigallocatechin gallate |
IC 50: 0.2 microM |
|
1.3.1.9 | (-)-gallocatechin gallate |
IC50: 0.5 microM |
|
1.3.1.9 | (1H-indol-5-yl)[4-[(4-methylphenyl)(phenyl)methyl]piperazin-1-yl]methanone |
0.015 mM, 74% inhibition |
|
1.3.1.9 | (2E)-1-[4-(1H-pyrrol-1-yl)phenyl]-3-[4-(trifluoromethyl)phenyl]prop-2-en-1-one |
- |
|
1.3.1.9 | (2E)-3-(1,2,3,4,5,6-hexahydropyrido[2,3-b][1,5]diazocin-8-yl)-N-methyl-N-[(3-methyl-1-benzofuran-2-yl)methyl]prop-2-enamide |
- |
|
1.3.1.9 | (2E)-3-(4-methoxyphenyl)-1-[4-(1H-pyrrol-1-yl)phenyl]prop-2-en-1-one |
- |
|
1.3.1.9 | (2E)-3-(4-methylphenyl)-1-[4-(1H-pyrrol-1-yl)phenyl]prop-2-en-1-one |
- |
|
1.3.1.9 | (2E)-3-(6-aminopyridin-3-yl)-N-(4-methoxyphenyl)prop-2-enamide |
- |
|