EC Number |
Inhibitors |
Structure |
---|
2.1.1.6 | (-)-epigallocatechin-3-gallate-7-O-glucuronide |
IC50: 600 nM with 2-hydroxyestradiol as substrate, IC50: 800 nM with 4-hydroxyestradiol as substrate |
|
2.1.1.6 | (-)-epigallocatechin-3-O-gallate |
IC50: 0.05-0.07 nM for the O-methylation of 2-hydroxyestradiol, IC50: 200-500 nM for O-methylation of 4-hydroxyestradiol |
|
2.1.1.6 | (-)-epigallocatechin-3-O-gallate |
potent non-competitive inhibitor |
|
2.1.1.6 | (-)-epigallocatechin-3-O-gallate |
- |
|
2.1.1.6 | (-)epicatechin |
IC50: 0.06 mM with 2-hydroxyestradiol as substrate, IC50: 0.08 mM with 4-hydroxyestradiol as substrate |
|
2.1.1.6 | (-)epicatechin gallate3,5-dinitrocatechol |
with epigallocatechin or 3,4-dihydroxy-L-Phe as substrates |
|
2.1.1.6 | (2-amino-3-methylbutanoyloxy)methyl-3-chloro-5,6-dihydroxy-7-nitrobenzo[b]thiophene-2-carboxylate |
- |
|
2.1.1.6 | (2E)-4,7-anhydro-1,2,3-trideoxy-1-(2,3-dihydroxy-5-nitrobenzamido)-L-ribo-hept-2-enitol |
- |
|
2.1.1.6 | (2R,3R)-5,7-bis(acetyloxy)-2-[3,4,5-tris(acetyloxy)phenyl]-3,4-dihydro-2H-chromen-3-yl 3,4-bis(acetyloxy)-5-(2-oxopropyl)benzoate |
- |
|
2.1.1.6 | (2R,3S)-1,2,3,4-tetrahydronaphthalene-2,3-diyl bis(3,4,5-trihydroxybenzoate) |
- |
|