Cloned (Comment) | Organism |
---|---|
expressed in Pichia pastoris | Mus musculus |
Crystallization (Comment) | Organism |
---|---|
hanging drop vapor diffusion method, using 100 mM HEPES, pH 7.5, 200 mM NaCl, 25% (w/v) PEG400 | Mus musculus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
elacridar | - |
Mus musculus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + H2O + xenobiotic[side 1] | Mus musculus | - |
ADP + phosphate + xenobiotic[side 2] | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Mus musculus | P21447 | - |
- |
Purification (Comment) | Organism |
---|---|
Ni-NTA column chromatography and Superdex 200 gel filtration | Mus musculus |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + H2O + calcein[side 1] | - |
Mus musculus | ADP + phosphate + calcein[side 2] | - |
? | |
ATP + H2O + cyclosporine A[side 1] | - |
Mus musculus | ADP + phosphate + cyclosporine A[side 2] | - |
? | |
ATP + H2O + quinidine[side 1] | - |
Mus musculus | ADP + phosphate + quinidine[side 2] | - |
? | |
ATP + H2O + rhodamine 123[side 1] | - |
Mus musculus | ADP + phosphate + rhodamine 123[side 2] | - |
? | |
ATP + H2O + verapamil[side 1] | - |
Mus musculus | ADP + phosphate + verapamil[side 2] | - |
? | |
ATP + H2O + xenobiotic[side 1] | - |
Mus musculus | ADP + phosphate + xenobiotic[side 2] | - |
? |
Subunits | Comment | Organism |
---|---|---|
? | x * 100000, SDS-PAGE | Mus musculus |
Synonyms | Comment | Organism |
---|---|---|
multidrug transporter | - |
Mus musculus |
P-glycoprotein | - |
Mus musculus |
P-gp | - |
Mus musculus |
Temperature Stability Minimum [°C] | Temperature Stability Maximum [°C] | Comment | Organism |
---|---|---|---|
42.5 | - |
melting temperature | Mus musculus |