Cloned (Comment) | Organism |
---|---|
expressed in Sf9 insect cells | Homo sapiens |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
membrane | - |
Homo sapiens | 16020 | - |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + H2O + xenobiotic[side 1] | Homo sapiens | - |
ADP + phosphate + xenobiotic[side 2] | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | Q9UNQ0 | - |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
breast cancer cell | - |
Homo sapiens | - |
duodenum | - |
Homo sapiens | - |
epithelial cell | - |
Homo sapiens | - |
gastrointestinal tract | - |
Homo sapiens | - |
kidney | - |
Homo sapiens | - |
liver | - |
Homo sapiens | - |
mammary gland | - |
Homo sapiens | - |
placenta | - |
Homo sapiens | - |
renal proximal tubule epithelial cell | - |
Homo sapiens | - |
syncytiotrophoblast | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + H2O + 2-amino-1-methyl-6-phenylimidazo[4,5-b]pyridine[side 1] | - |
Homo sapiens | ADP + phosphate + 2-amino-1-methyl-6-phenylimidazo[4,5-b]pyridine[side 2] | - |
? | |
ATP + H2O + cimetidine[side 1] | - |
Homo sapiens | ADP + phosphate + cimetidine[side 2] | - |
? | |
ATP + H2O + daunomycin[side 1] | - |
Homo sapiens | ADP + phosphate + daunomycin[side 2] | - |
? | |
ATP + H2O + daunorubicin[side 1] | - |
Homo sapiens | ADP + phosphate + daunorubicin[side 2] | - |
? | |
ATP + H2O + doxorubicin[side 1] | - |
Homo sapiens | ADP + phosphate + doxorubicin[side 2] | - |
? | |
ATP + H2O + Hoechst 33342[side 1] | - |
Homo sapiens | ADP + phosphate + Hoechst 33342[side 2] | - |
? | |
ATP + H2O + lyso-tracker green[side 1] | - |
Homo sapiens | ADP + phosphate + lyso-tracker green[side 2] | - |
? | |
ATP + H2O + methotrexate[side 1] | - |
Homo sapiens | ADP + phosphate + methotrexate[side 2] | - |
? | |
ATP + H2O + mitoxantrone[side 1] | - |
Homo sapiens | ADP + phosphate + mitoxantrone[side 2] | - |
? | |
ATP + H2O + prazosin[side 1] | - |
Homo sapiens | ADP + phosphate + prazosin[side 2] | - |
? | |
ATP + H2O + rhodamine 123[side 1] | - |
Homo sapiens | ADP + phosphate + rhodamine 123[side 2] | - |
? | |
ATP + H2O + riboflavin[side 1] | - |
Homo sapiens | ADP + phosphate + riboflavin[side 2] | - |
? | |
ATP + H2O + topotecan[side 1] | - |
Homo sapiens | ADP + phosphate + topotecan[side 2] | - |
? | |
ATP + H2O + xenobiotic[side 1] | - |
Homo sapiens | ADP + phosphate + xenobiotic[side 2] | - |
? |
Synonyms | Comment | Organism |
---|---|---|
ABCG2 | - |
Homo sapiens |
breast cancer resistance protein | - |
Homo sapiens |
multidrug transporter | - |
Homo sapiens |
General Information | Comment | Organism |
---|---|---|
physiological function | the localization of enzyme ABCG2 can play a vital role in limiting absorption (in the small intestine), mediating distribution (e.g. in the blood-brain and blood-placental barriers) and facilitating elimination and excretion (in the liver and kidney) of drugs or xenobiotics | Homo sapiens |