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BRENDA support

Literature summary for 5.6.2.2 extracted from

  • Vosberg, H.P.
    Topoisomerasen und Gyrasehemmer (1986), Fortschr. Antimikrob. Antiplast. Chemother., 5, 761-767.
No PubMed abstract available

Inhibitors

Inhibitors Comment Organism Structure
coumermycin
-
Escherichia coli
doxorubicin
-
Escherichia coli
Nalidixic acid
-
Bacteria
Nalidixic acid
-
Escherichia coli
novobiocin
-
Bacteria
novobiocin
-
Escherichia coli
Oxolinic acid
-
Bacteria
Oxolinic acid
-
Escherichia coli

Molecular Weight [Da]

Molecular Weight [Da] Molecular Weight Maximum [Da] Comment Organism
400000
-
-
Escherichia coli

Organism

Organism UniProt Comment Textmining
Bacteria
-
-
-
Escherichia coli
-
-
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
network of DNA rings + ATP + H2O decatenation Bacteria monomeric DNA circles + ADP + phosphate
-
?
network of DNA rings + ATP + H2O decatenation Escherichia coli monomeric DNA circles + ADP + phosphate
-
?
supercoiled DNA + ATP + H2O catenation Bacteria catenated DNA networks + ADP + phosphate
-
?
supercoiled DNA + ATP + H2O catenation Escherichia coli catenated DNA networks + ADP + phosphate
-
?
supercoiled DNA + ATP + H2O relaxation Bacteria relaxed DNA + ADP + phosphate
-
?
supercoiled DNA + ATP + H2O relaxation Escherichia coli relaxed DNA + ADP + phosphate
-
?
supercoiled DNA + ATP + H2O relaxation of negatively or positively supercoiled DNA Bacteria relaxed DNA + ADP + phosphate
-
?
supercoiled DNA + ATP + H2O relaxation of negatively or positively supercoiled DNA Escherichia coli relaxed DNA + ADP + phosphate
-
?