Cloned (Comment) | Organism |
---|---|
expression in Escherichia coli | Plasmodium falciparum |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
methylglutathione | - |
Plasmodium falciparum | |
S-nitrosoglutathione | - |
Plasmodium falciparum | |
S-p-nitrosobenzylglutathione | - |
Plasmodium falciparum |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.077 | - |
glutathione-methylglyoxal hemithioacetal | - |
Plasmodium falciparum | |
0.58 | - |
glutathione-glyoxal hemithioacetal | - |
Plasmodium falciparum |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Ni2+ | 2.9fold increase in activity at 0.25 mM | Plasmodium falciparum | |
Zn2+ | 2.7fold increase in activity at 0.25 mM | Plasmodium falciparum |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
42300 | - |
gel filtration | Plasmodium falciparum |
43600 | - |
1 * 43600, SDS-PAGE, recombinant His-tagged PfGlx I | Plasmodium falciparum |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
glutathione-glyoxal hemithioacetal | Plasmodium falciparum | - |
? | - |
? | |
glutathione-methylglyoxal hemithioacetal | Plasmodium falciparum | glutathione-methylglyoxal hemithioacetal is formed non-enzymatically from methylglyoxal and glutathione | (R)-S-lactoylglutathione | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Plasmodium falciparum | Q71KM3 | - |
- |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
90 | - |
- |
Plasmodium falciparum |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
glutathione-glyoxal hemithioacetal | - |
Plasmodium falciparum | ? | - |
? | |
glutathione-methylglyoxal hemithioacetal | glutathione-methylglyoxal hemithioacetal is formed non-enzymatically from methylglyoxal and glutathione | Plasmodium falciparum | (R)-S-lactoylglutathione | - |
? |
Subunits | Comment | Organism |
---|---|---|
monomer | 1 * 43600, SDS-PAGE, recombinant His-tagged PfGlx I | Plasmodium falciparum |
Synonyms | Comment | Organism |
---|---|---|
glyoxalase I | - |
Plasmodium falciparum |
PfGlx I | - |
Plasmodium falciparum |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
66.7 | - |
glutathione-methylglyoxal hemithioacetal | - |
Plasmodium falciparum |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.8 | - |
- |
Plasmodium falciparum |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.06 | - |
S-p-nitrosobenzylglutathione | - |
Plasmodium falciparum | |
0.17 | - |
methylglutathione | - |
Plasmodium falciparum | |
0.19 | - |
S-p-nitrosobenzylglutathione | - |
Plasmodium falciparum |