General Stability | Organism |
---|---|
proteolytic cleavage at Arg330 and subsequent inactivation can be diminished by the addition of 6-aminohexanoic acid, 5-aminopentanoic acid, 7-aminoheptanoic acid, hippuryl-L-Lys, hippuryl-L-Arg, L-Arg, or L-Lys | Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
10 | - |
bradykinin | - |
Homo sapiens | |
63 | - |
Arg6-Leu5-enkephalin | - |
Homo sapiens | |
110 | - |
Lys6-Leu5-enkephalin | - |
Homo sapiens | |
140 | - |
Arg6-Met5-enkephalin | - |
Homo sapiens | |
180 | - |
hippuryl-L-Arg | - |
Homo sapiens | |
210 | - |
N-[3-(2-Furylacryloyl)]-L-Ala-L-Arg | - |
Homo sapiens | |
220 | - |
Lys6-Met5-enkephalin | - |
Homo sapiens | |
240 | - |
Hippuryl-L-argininic acid | - |
Homo sapiens | |
270 | - |
Hippuryl-L-Lys | - |
Homo sapiens | |
280 | - |
N-[3-(2-Furylacryloyl)]-L-Ala-L-Lys | - |
Homo sapiens |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Zn2+ | metalloproteinase | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
plasma | - |
Homo sapiens | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
additional information | - |
- |
Homo sapiens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
Arg6-Leu5-enkephalin + H2O | i.e. Tyr-Gly-Gly-Phe-Leu-Arg | Homo sapiens | Tyr-Gly-Gly-Phe-Leu + Arg | - |
? | |
Arg6-Met5-enkephalin + H2O | i.e. Tyr-Gly-Gly-Phe-Met-Arg | Homo sapiens | Tyr-Gly-Gly-Phe-Met + Arg | - |
? | |
bradykinin + H2O | i.e. Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg | Homo sapiens | Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe + Arg | - |
? | |
Hippuryl-L-Arg + H2O | - |
Homo sapiens | Hippuric acid + L-Arg | - |
? | |
Hippuryl-L-argininic acid + H2O | - |
Homo sapiens | Hippuric acid + argininic acid | - |
? | |
Hippuryl-L-Lys + H2O | - |
Homo sapiens | Hippuric acid + L-Lys | - |
? | |
Lys6-Leu5-enkephalin + H2O | i.e. Tyr-Gly-Gly-Phe-Leu-Lys | Homo sapiens | Tyr-Gly-Gly-Phe-Leu + Lys | - |
? | |
Lys6-Met5-enkephalin + H2O | i.e. Tyr-Gly-Gly-Phe-Met-Lys | Homo sapiens | Tyr-Gly-Gly-Phe-Met + Lys | - |
? | |
N-[3-(2-Furylacryloyl)]-L-Ala-L-Arg + H2O | - |
Homo sapiens | N-[3-(2-Furylacryloyl)]-L-Ala + L-Arg | - |
? | |
N-[3-(2-Furylacryloyl)]-L-Ala-L-Lys + H2O | - |
Homo sapiens | N-[3-(2-Furylacryloyl)]-L-Ala + L-Lys | - |
? |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
15 | - |
Hippuryl-L-Lys | - |
Homo sapiens | |
26 | - |
hippuryl-L-Arg | - |
Homo sapiens | |
29 | - |
N-[3-(2-Furylacryloyl)]-L-Ala-L-Lys | - |
Homo sapiens | |
36 | - |
N-[3-(2-Furylacryloyl)]-L-Ala-L-Arg | - |
Homo sapiens | |
121 | - |
bradykinin | - |
Homo sapiens | |
169 | - |
Hippuryl-L-argininic acid | - |
Homo sapiens | |
282 | - |
Lys6-Leu5-enkephalin | - |
Homo sapiens | |
290 | - |
Lys6-Met5-enkephalin | - |
Homo sapiens | |
647 | - |
Arg6-Met5-enkephalin | - |
Homo sapiens | |
748 | - |
Arg6-Leu5-enkephalin | - |
Homo sapiens |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.5 | 9 | ester substrates | Homo sapiens |
7.5 | 8 | peptide substrates | Homo sapiens |