Activating Compound | Comment | Organism | Structure |
---|---|---|---|
diacylglycerol | - |
Rattus norvegicus | |
mezerein | stimulates classical, but not novel PKC isozymes | Rattus norvegicus | |
phorbol 12,13-dibutyrate | activates PKC, activates Na+,K+-ATPase activity at low concentration, but inhibits it at high concentration | Rattus norvegicus | |
phorbol 12-myristate 13-acetate | - |
Rattus norvegicus | |
thymeleatoxin | activates Na+,K+-ATPase activity at low concentration, but inhibits it at high concentration | Rattus norvegicus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
GF109203X | inhibits classical and novel, but not atypical PKC isozymes | Rattus norvegicus | |
GΓΆ-6976 | inhibits classical, but not novel and atypical PKC isozymes | Rattus norvegicus | |
LY333531 | specific inhibition of PKCbeta | Rattus norvegicus | |
phorbol 12,13-dibutyrate | activates Na+,K+-ATPase activity at low concentration, but inhibits it at high concentration, the inhibitory effect can be reversed by preincubation with ethoxyresorufin, 17-octadecynoic acid, wortmannin, LY294002, cytochlasin D, or latrunculin B | Rattus norvegicus | |
staurosporine | inhibits all PKC isozymes | Rattus norvegicus | |
thymeleatoxin | activates Na+,K+-ATPase activity at low concentration, but inhibits it at high concentration | Rattus norvegicus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
additional information | Rattus norvegicus | bidirectional regulation of renal cortical Na+,K+-ATPase by PKC | ? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Rattus norvegicus | - |
male Wistar rats | - |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
kidney | - |
Rattus norvegicus | - |
renal cortex | - |
Rattus norvegicus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
additional information | bidirectional regulation of renal cortical Na+,K+-ATPase by PKC | Rattus norvegicus | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
PKC | - |
Rattus norvegicus |