EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   3.4.21.26 | -999 |
- |
more |
- |
683553 |
| 3.4.21.26 | 0.000000023 |
- |
(2S)-1-[1-(4-phenylbutanoyl)-L-prolyl]pyrrolidine-2-carbonitrile |
- |
709476 |
| 3.4.21.26 | 0.00000015 |
- |
4-phenylbutanoyl-5(R)-methyl-L-Pro-2(S)-(hydroxyacetyl)pyrrolidine |
IC50: 0.15 nM |
650529 |
| 3.4.21.26 | 0.00000015 |
- |
KYP-2047 |
wild type enzyme, at pH 8.0 and 25°C |
731346 |
| 3.4.21.26 | 0.0000002 |
- |
4-phenylbutanoyl-L-prolyl-2(S)-(hydroxyacetyl)pyrrolidine |
IC50: 0.2 nM |
650521 |
| 3.4.21.26 | 0.0000002 |
- |
4-phenylbutanoyl-L-prolyl-2(S)-cyanopyrrolidine |
at 25°C between pH 5.5 and 9.5 |
731374 |
| 3.4.21.26 | 0.0000002 |
- |
JTP-4819 |
IC50: 0.2 nM |
650521 |
| 3.4.21.26 | 0.00000024 |
- |
4-phenylbutanoyl-L-Pro-2(S)-(hydroxyacetyl)-pyrrolidine |
IC50: 0.24 nM |
650529 |
| 3.4.21.26 | 0.00000026 |
- |
4-phenylbutanoyl-5(R)-tert-butyl-L-Pro-2(S)-(hydroxyacetyl)-pyrrolidine |
IC50: 0.26 nM |
650529 |
| 3.4.21.26 | 0.00000026 |
- |
4-phenylbutanoyl-5(R)-tert-butyl-L-prolyl-2(S)-(hydroxyacetyl)pyrrolidine |
at 25°C between pH 5.5 and 9.5 |
731374 |
