EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.3.3.4 | -999 |
- |
more |
pI50 values of 3H-pyrazolo[3,4-d][1,2,3]triazin-4-one derivative inhibitors, overview |
699636 |
1.3.3.4 | -999 |
- |
more |
pI50 values of H-pyrazolo[3,4-d][1,2,3]triazin-4-one derivative inhibitors, overview |
698439 |
1.3.3.4 | 0.0000012 |
- |
2-chloroethyl 2-[[([2-chloro-4-fluoro-5-[3-methyl-2,6-dioxo-4-(trifluoromethyl)-3,6-dihydropyrimidin-1(2H)-yl]phenyl]amino)methyl]sulfanyl]propanoate |
pH and temperature not specified in the publication |
764962 |
1.3.3.4 | 0.0000023 |
- |
ethyl 2-[[([2-chloro-4-fluoro-5-[3-methyl-2,6-dioxo-4-(trifluoromethyl)-3,6-dihydropyrimidin-1(2H)-yl]phenyl]amino)methyl]sulfanyl]propanoate |
pH and temperature not specified in the publication |
764962 |
1.3.3.4 | 0.0000026 |
- |
2-[[([2-chloro-4-fluoro-5-[3-methyl-2,6-dioxo-4-(trifluoromethyl)-3,6-dihydropyrimidin-1(2H)-yl]phenyl]amino)methyl]sulfanyl]-N-ethylpropanamide |
pH and temperature not specified in the publication |
764962 |
1.3.3.4 | 0.000003 |
- |
2-[[([2-chloro-4-fluoro-5-[3-methyl-2,6-dioxo-4-(trifluoromethyl)-3,6-dihydropyrimidin-1(2H)-yl]phenyl]amino)methyl]sulfanyl]-N-propylacetamide |
pH and temperature not specified in the publication |
764962 |
1.3.3.4 | 0.0000036 |
- |
2-[[([2-chloro-4-fluoro-5-[3-methyl-2,6-dioxo-4-(trifluoromethyl)-3,6-dihydropyrimidin-1(2H)-yl]phenyl]amino)methyl]sulfanyl]-N-ethylacetamide |
pH and temperature not specified in the publication |
764962 |
1.3.3.4 | 0.000004 |
- |
1-(tert-butoxy)-1-oxopropan-2-yl 2-chloro-4-fluoro-5-(4-oxo-5,6,7,8-tetrahydroquinazolin-3(4H)-yl)benzoate |
pH and temperature not specified in the publication |
764284 |
1.3.3.4 | 0.0000044 |
- |
2-ethoxy-2-oxoethyl [([2-chloro-4-fluoro-5-[3-methyl-2,6-dioxo-4-(trifluoromethyl)-3,6-dihydropyrimidin-1(2H)-yl]anilino]methyl)sulfanyl]acetate |
pH and temperature not specified in the publication |
764962 |
1.3.3.4 | 0.0000046 |
- |
ethyl 3-[2-chloro-4-fluoro-5-(1-oxo-3-thioxotetrahydro-1H-[1,2,4]triazolo[1,2-a]pyridazin-2(3H)-yl)phenyl]-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate |
at pH 7.4, temperature not specified in the publication |
764954 |