EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.6.1.27 | 0.00003 |
0.0001 |
tripropeptin C |
in 100 mM Tris-HCl, 10 mM MgCl2 and 3.9 mM n-dodecyl-beta-maltoside (pH 7.5), 1.25 mM CaCl2, at 30°C |
718588 |
3.6.1.27 | 0.00083 |
- |
2-[3-(octyloxy)benzamido]-5-(trifluoromethoxy)benzoic acid |
at pH 7.5 and 20°C |
756478 |
3.6.1.27 | 0.00083 |
- |
2-[3-(octyloxy)benzamido]-5-(trifluoromethoxy)benzoic acid |
pH and temperature not specified in the publication, mutant enzyme Y246D |
756478 |
3.6.1.27 | 0.0013 |
- |
5-fluoro-2-[3-(octyloxy)benzamido]benzoic acid |
pH and temperature not specified in the publication, mutant enzyme Y246D |
756478 |
3.6.1.27 | 0.0013 |
- |
5-nitro-2-[3-(octyloxy)benzamido]benzoic acid |
at pH 7.5 and 20°C |
756478 |
3.6.1.27 | 0.0027 |
- |
5-fluoro-2-(3-(octyloxy)benzamido)benzoic acid |
at pH 7.5 and 20°C |
756478 |
3.6.1.27 | 0.0027 |
- |
5-fluoro-2-[3-(octyloxy)benzamido]benzoic acid |
pH and temperature not specified in the publication, mutant enzyme Y246D |
756478 |
3.6.1.27 | 0.003 |
- |
5-chloro-2-[3-(octyloxy)benzamido]benzoic acid |
at pH 7.5 and 20°C |
756478 |
3.6.1.27 | 0.003 |
- |
5-chloro-2-[3-(octyloxy)benzamido]benzoic acid |
pH and temperature not specified in the publication, mutant enzyme Y246D |
756478 |
3.6.1.27 | 0.0034 |
- |
4,5-difluoro-2-[3-(octyloxy)benzamido]benzoic acid |
at pH 7.5 and 20°C |
756478 |