EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   3.4.21.B28 | 0.0000033 |
- |
N-[2-(2-cyano-4,4-difluoropyrrolidin-1-yl)-2-oxoethyl]quinoline-4-carboxamide |
pH and temperature not specified in the publication |
732455 |
| 3.4.21.B28 | 0.00004 |
- |
Talabostat |
- |
678473 |
| 3.4.21.B28 | 0.00007 |
- |
[(2S)-1-(D-valyl)pyrrolidin-2-yl]boronic acid |
pH and temperature not specified in the publication |
732455 |
| 3.4.21.B28 | 0.000089 |
0.00037 |
linagliptin |
pH and temperature not specified in the publication |
732455 |
| 3.4.21.B28 | 0.00074 |
- |
7-(but-2-yn-1-yl)-3-methyl-1-[(4-methylquinazolin-2-yl)methyl]-8-(piperazin-1-yl)-3,7-dihydro-1H-purine-2,6-dione |
pH and temperature not specified in the publication |
732455 |
| 3.4.21.B28 | 0.0012 |
- |
7-(but-2-yn-1-yl)-1-[(4-methoxyquinazolin-2-yl)methyl]-3-methyl-8-(piperazin-1-yl)-3,7-dihydro-1H-purine-2,6-dione |
pH and temperature not specified in the publication |
732455 |
| 3.4.21.B28 | 0.0018 |
- |
7-(but-2-yn-1-yl)-3-methyl-8-(piperazin-1-yl)-1-(quinazolin-2-ylmethyl)-3,7-dihydro-1H-purine-2,6-dione |
pH and temperature not specified in the publication |
732455 |
| 3.4.21.B28 | 0.0019 |
- |
7-(but-2-yn-1-yl)-3-methyl-1-[(4-methylquinazolin-2-yl)methyl]-8-(3-oxopiperazin-1-yl)-3,7-dihydro-1H-purine-2,6-dione |
pH and temperature not specified in the publication |
732455 |
| 3.4.21.B28 | 0.0026 |
- |
saxagliptin |
pH and temperature not specified in the publication |
732455 |
| 3.4.21.B28 | 0.0033 |
- |
7-(but-2-yn-1-yl)-8-[(3S)-3-(hydroxymethyl)-5-oxopiperazin-1-yl]-3-methyl-1-[(4-methylquinazolin-2-yl)methyl]-3,7-dihydro-1H-purine-2,6-dione |
pH and temperature not specified in the publication |
732455 |
